SCHEMBL4949101

SCHEMBL4949101

Cc1cc(S(C)(=O)=O)c2ncc(C(N)=O)c(Nc3cccc4c3CCO4)c2c1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.68
MTNR1B P49286 1/20 0.39
CSF1R P07333 4/20 0.38
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4952737 0.95 PDE4B (0.61) PDE4BCSF1RTHRB
SCHEMBL4949456 0.91 PDE4B (0.67) PDE4BMTNR1BCSF1R
SCHEMBL4950089 0.91 PDE4B (0.67) PDE4BMTNR1BCSF1R
SCHEMBL4949711 0.90 PDE4B (0.64) PDE4BMTNR1BCSF1R
SCHEMBL4949173 0.89 PDE4B (0.69) PDE4BMTNR1BCSF1R
SCHEMBL4951313 0.89 PDE4B (0.65) PDE4BMTNR1BCSF1R
SCHEMBL4945356 0.88 PDE4B (0.58) PDE4BMTNR1BCSF1RTHRB
SCHEMBL4628322 0.88 PDE4B (0.57) PDE4BMTNR1BCSF1R
SCHEMBL8311654 0.87 PDE4B (0.66) PDE4BMTNR1BCSF1R
SCHEMBL4949741 0.87 PDE4B (0.60) PDE4BCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed