SCHEMBL4949063

SCHEMBL4949063

Cc1cc(S(C)(=O)=O)c2ncc(C(N)=O)c(Nc3cccc(F)c3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 6/20 0.56
PDE4B Q07343 13/20 0.54
LMNA P02545 1/20 0.47
LRRK2 Q5S007 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4948831 0.90 PDE4B (0.56) CSF1RPDE4BLMNALRRK2
SCHEMBL4951564 0.90 CSF1R (0.53) CSF1RPDE4BLRRK2
SCHEMBL4948930 0.88 CSF1R (0.53) CSF1RPDE4BLMNALRRK2
SCHEMBL4952739 0.87 PDE4B (0.48) CSF1RPDE4BLRRK2
SCHEMBL4952577 0.86 PDE4B (0.74) CSF1RPDE4BLRRK2
SCHEMBL4951405 0.85 PDE4B (0.63) CSF1RPDE4BLRRK2
SCHEMBL4949236 0.85 PDE4B (0.66) CSF1RPDE4B
SCHEMBL1276135 0.84 PDE4B (0.75) CSF1RPDE4BLRRK2
SCHEMBL4948799 0.84 PDE4B (0.56) CSF1RPDE4BLRRK2
SCHEMBL4627712 0.84 PDE4B (0.54) CSF1RPDE4BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed