SCHEMBL4948854

SCHEMBL4948854

Cc1cc(S(C)(=O)=O)c2ncc(C(N)=O)c(Nc3cccc(F)c3F)c2c1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 10/20 0.56
PDE4B Q07343 6/20 0.54
JAK2 O60674 1/20 0.43
JAK1 P23458 1/20 0.43
TYK2 P29597 1/20 0.43
JAK3 P52333 1/20 0.43
BRD4 O60885 1/20 0.43
BRD2 P25440 1/20 0.43
BRD3 Q15059 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4944374 0.91 PDE4B (0.67) CSF1RPDE4BJAK2JAK1TYK2
SCHEMBL1276139 0.85 PDE4B (0.65) CSF1RPDE4B
SCHEMBL4949063 0.83 CSF1R (0.56) CSF1RPDE4B
SCHEMBL4951564 0.81 CSF1R (0.53) CSF1RPDE4B
SCHEMBL4949101 0.80 PDE4B (0.68) CSF1RPDE4B
SCHEMBL4952737 0.79 PDE4B (0.61) CSF1RPDE4B
SCHEMBL4952739 0.78 PDE4B (0.48) CSF1RPDE4B
SCHEMBL4951405 0.78 PDE4B (0.63) CSF1RPDE4B
SCHEMBL4952577 0.77 PDE4B (0.74) CSF1RPDE4B
SCHEMBL4951019 0.77 PDE4B (0.46) CSF1RPDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed