SCHEMBL4947199

SCHEMBL4947199

CC(NC(=O)C(O)c1cc(F)cc(F)c1)C(=O)Nc1cc(C(C)Cc2cccc(C(F)(F)F)c2)n[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.44
MMP2 P08253 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
PSEN1 P49768 5/20 0.37
PSEN2 P49810 5/20 0.37
APH1B Q8WW43 5/20 0.37
NCSTN Q92542 5/20 0.37
APH1A Q96BI3 5/20 0.37
PSENEN Q9NZ42 5/20 0.37
KCNJ6 P48051 1/20 0.36
KCNJ5 P48544 1/20 0.36
KCNJ3 P48549 1/20 0.36
HTR2A P28223 3/20 0.36
HTR2B P41595 3/20 0.36
HTR2C P28335 2/20 0.36
ADRA2C P18825 2/20 0.35
SLC6A4 P31645 2/20 0.35
ADRA1A P35348 2/20 0.35
DRD3 P35462 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2956970 0.91 PSEN1 (0.40) MMP1MMP2MMP9MMP8PSEN1
SCHEMBL4945243 0.89 PSEN1 (0.43) MMP1MMP2MMP9MMP8PSEN1
SCHEMBL4947202 0.84 MMP1 (0.41) MMP1MMP2MMP9MMP8PSEN1
SCHEMBL8313682 0.81 PSEN1 (0.38) MMP1MMP2MMP9MMP8PSEN1
SCHEMBL2958410 0.81 PSEN1 (0.38) MMP1MMP2MMP9MMP8PSEN1
SCHEMBL4942350 0.80 MMP2 (0.42) MMP1MMP2MMP9MMP8
SCHEMBL2968170 0.79 MMP1 (0.36) MMP1MMP2MMP9MMP8PSEN1
SCHEMBL8322329 0.78 PSEN1 (0.45) MMP1MMP2MMP9MMP8PSEN1
SCHEMBL8322384 0.78 PSEN1 (0.43) MMP1MMP2MMP9MMP8PSEN1
SCHEMBL2965388 0.78 PSEN1 (0.43) MMP1MMP2MMP9MMP8PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633350-A4 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS ELAN PHARM INC (US) 2008-11-26 EP disclosed
EP-1633350-A2 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS Elan Pharmaceuticals, Inc. (US) 2006-03-15 EP disclosed
WO-2005009344-A2 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 2005-02-03 WO disclosed