SCHEMBL4948050

SCHEMBL4948050

CC(C)(C)OC(=O)N(C(=O)OC(C)(C)C)c1nc2cc(Cl)c([N+](=O)[O-])cc2n1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
PGK1 P00558 1/20 0.35
EGLN1 Q9GZT9 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPT P10636 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MET P08581 1/20 0.32
HPGD P15428 1/20 0.31
SLC9A1 P19634 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
GPR55 Q9Y2T6 1/20 0.31
CA12 O43570 1/20 0.31
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4089267 0.92 LMNA (0.38) LMNAPGK1EGLN1ALDH1A1MAPT
SCHEMBL4946449 0.83 KDM4E (0.31) ALDH1A1MAPTNPC1RAB9AHPGD
SCHEMBL4091251 0.74 AURKA (0.35) MAPTNPC1RAB9A
SCHEMBL482970 0.73 BACE1 (0.35) ALDH1A1MAPTNPC1RAB9A
SCHEMBL18459405 0.72 BRD4 (0.42) LMNAALDH1A1MAPTNPC1RAB9A
SCHEMBL3100964 0.72 ALDH1A1 (0.38) LMNAALDH1A1MAPTHPGDCYP1A2
SCHEMBL481938 0.72
SCHEMBL27851953 0.70 L3MBTL1 (0.35) ALDH1A1MAPTNPC1RAB9A
SCHEMBL30628499 0.69 MAPT (0.36) LMNAALDH1A1MAPTMETHPGD
SCHEMBL26632138 0.69 MAPT (0.34) LMNAALDH1A1MAPTMETHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885362-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-02-13 EP disclosed
WO-2006127458-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-30 WO disclosed