SCHEMBL4948136

SCHEMBL4948136

Nc1nc(Nc2cccc(O)c2)nc2c1ncn2CCOCP

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 1/20 0.44
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
ADORA2A P29274 5/20 0.41
TMIGD3 P0DMS9 4/20 0.41
ADORA1 P30542 4/20 0.41
ADORA2B P29275 3/20 0.40
CYP1A2 P05177 2/20 0.38
KMT2A Q03164 2/20 0.38
THPO P40225 1/20 0.38
MEN1 O00255 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
BLM P54132 1/20 0.38
SYK P43405 2/20 0.37
FGFR1 P11362 1/20 0.36
SLC22A6 Q4U2R8 1/20 0.36
CDK1 P06493 2/20 0.35
CHKA P35790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12396113 0.79 TMIGD3 (0.41) PDGFRACCNE1CDK2ADORA2ATMIGD3
SCHEMBL215612 0.73 CDK1 (0.57) CCNE1CDK2FGFR1SLC22A6CDK1
SCHEMBL4948978 0.69 CYP1A2 (0.49) ADORA2AADORA2BCYP1A2KMT2ATHPO
SCHEMBL4948967 0.69 CYP1A2 (0.49) ADORA2AADORA2BCYP1A2KMT2ATHPO
SCHEMBL2160243 0.68 FGFR1 (0.47) PDGFRACCNE1CDK2ADORA2ATMIGD3
SCHEMBL8154514 0.67 ADORA2A (0.43) ADORA2ATMIGD3ADORA1ADORA2BCYP1A2
SCHEMBL4949185 0.67 CYP1A2 (0.47) PDGFRACCNE1CDK2ADORA2AADORA2B
SCHEMBL4949178 0.67 CYP1A2 (0.47) PDGFRACCNE1CDK2ADORA2AADORA2B
SCHEMBL7209426 0.67 PDE4A (0.60) PDGFRACCNE1CDK2ADORA2ATMIGD3
SCHEMBL382916 0.67 FGFR1 (0.66) ADORA2AADORA1ADORA2BFGFR1SLC22A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1990054-A1 Polymerase inhibitors and their use in treating tumours Freie Universität Berlin (DE) 2008-11-12 EP disclosed