SCHEMBL4948686

SCHEMBL4948686

NC(=O)CNCCCc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.62
L3MBTL1 Q9Y468 1/20 0.54
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
GAA P10253 1/20 0.53
HPGD P15428 1/20 0.53
FDPS P14324 1/20 0.53
EPHX2 P34913 1/20 0.51
LMNA P02545 1/20 0.50
KDM4E B2RXH2 1/20 0.50
EPHX1 P07099 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4953206 0.95 SIGMAR1 (0.61) SIGMAR1FDPS
SCHEMBL4344215 0.89 TAAR1 (0.54) SIGMAR1NPC1RAB9AGAAFDPS
SCHEMBL13469007 0.86 BCHE (0.67) SIGMAR1NPC1RAB9AEPHX2
SCHEMBL158734 0.85 SIGMAR1 (0.67) SIGMAR1L3MBTL1NPC1RAB9AGAA
SCHEMBL5106492 0.84 MAOB (0.46) SIGMAR1L3MBTL1FDPS
SCHEMBL5099654 0.84 CA2 (0.48) SIGMAR1L3MBTL1KDM4ECYP2C19
SCHEMBL10766680 0.84 SIGMAR1 (0.66) SIGMAR1L3MBTL1FDPS
SCHEMBL9776078 0.83 LMNA (0.47) SIGMAR1L3MBTL1NPC1RAB9AGAA
SCHEMBL9776115 0.83 LMNA (0.47) SIGMAR1L3MBTL1NPC1RAB9AGAA
SCHEMBL5106212 0.83 HDAC3 (0.46) SIGMAR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008026075-A2 TREATMENT OF INTRACELLULAR BACTERIAL INFECTIONS WITH A PROTEIN KINASE INHIBITOR OR AN AS160 POLYPEPTIDE ACTIVATOR VERENIGING HET NEDERLANDS KANKER INSTITUUT (NL) 2008-03-06 WO disclosed
US-6420385-B1 INFLAMMATORY, PAIN AND DIABETES DISEASES, AMGEN INC. 2002-07-16 US disclosed
US-5672615-A MATRIX-DEGRADING METALLOPROTEINASE INHIBITORS NOVARTIS CORPORATION (US) 1997-09-30 US disclosed
US-4639468-A Derivatives of glycinamide, their preparation and their use CONTINENTAL PHARMA INC. (BE) 1987-01-27 US disclosed