SCHEMBL4948723

SCHEMBL4948723

Nc1cccc(NS(=O)(=O)c2ccc([N+](=O)[O-])cc2)c1

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.72
CA2 P00918 3/20 0.68
CA12 O43570 1/20 0.68
CA9 Q16790 1/20 0.68
FFAR4 Q5NUL3 2/20 0.60
CA1 P00915 2/20 0.60
MAPT P10636 2/20 0.58
MAPK1 P28482 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58
LMNA P02545 1/20 0.58
POLB P06746 2/20 0.55
HTT P42858 1/20 0.54
PIK3CB P42338 1/20 0.52
ALDH1A1 P00352 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28506881 0.90 HTR6 (0.66) HTR6CA2CA12CA9FFAR4
Trifluoroacetic Acid SCHEMBL15648070 0.89 FFAR4 (0.59) HTR6CA2CA12CA9FFAR4
SCHEMBL1024534 0.89 ALDH1A1 (0.65) HTR6CA2FFAR4CA1KMT2A
SCHEMBL13265931 0.85 HTR6 (0.53) HTR6CA2CA12CA9FFAR4
SCHEMBL27888184 0.85 HTR6 (0.68) HTR6CA2CA12CA9FFAR4
SCHEMBL28271812 0.84 HTR6 (1.00) HTR6CA2CA9CA1KMT2A
SCHEMBL28271833 0.83 HTR6 (0.54) HTR6CA2CA12CA9FFAR4
SCHEMBL28270344 0.83 HTR6 (0.64) HTR6CA2CA12CA9FFAR4
SCHEMBL28270327 0.82 GUSB (0.56) HTR6CA2CA12CA9FFAR4
SCHEMBL2243550 0.82 CA2 (0.68) CA2CA12CA9FFAR4CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109081793-B Sulfonamide urease inhibitor and preparation method and application thereof 吉首大学 2021-03-30 CN disclosed
CN-109081793-A Sulfonamides urease inhibitor and its preparation method and purposes 吉首大学 2018-12-25 CN disclosed
CN-107810189-A Method for preparing nitrogen mustard derivatives 肿瘤多肽股份公司 2018-03-16 CN disclosed
EP-1218360-B1 TRIAZINE KINASE INHIBITORS AMGEN INC (US) 2008-05-28 EP disclosed
US-7074789-B2 Kinase inhibitors AMGEN INC. (US) 2006-07-11 US disclosed
EP-1218360-A1 TRIAZINE KINASE INHIBITORS Amgen Inc., (US) 2002-07-03 EP disclosed
WO-2001025220-A1 TRIAZINE KINASE INHIBITORS AMGEN INC. (US) 2001-04-12 WO disclosed