Glenvastatin

Glenvastatin

SCHEMBL49508

CC(C)c1nc(-c2ccccc2)cc(-c2ccc(F)cc2)c1/C=C/[C@@H]1C[C@@H](O)CC(=O)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 12/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Glenvastatin SCHEMBL1040745 1.00 HMGCR (1.00) HMGCR
Glenvastatin SCHEMBL29557142 1.00 HMGCR (1.00) HMGCR
Glenvastatin SCHEMBL1040744 1.00 HMGCR (1.00) HMGCR
Glenvastatin SCHEMBL9872411 1.00 HMGCR (1.00) HMGCR
SCHEMBL9022892 1.00 HMGCR (1.00) HMGCR
Glenvastatin SCHEMBL1660022 1.00 HMGCR (1.00) HMGCR
Glenvastatin SCHEMBL10024037 1.00 HMGCR (1.00) HMGCR
SCHEMBL9527887 0.96 HMGCR (1.00) HMGCR
SCHEMBL9022328 0.94 HMGCR (0.89) HMGCR
SCHEMBL9023237 0.92 HMGCR (0.85) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1315 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3875078-A1 COMPOUNDS FOR THE TREATMENT OF COVID-19 Dompe' Farmaceutici S.P.A. (IT) 2021-09-08 EP claimed
US-20210085695-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF MIGRAINE HEADACHES BETH ISRAEL DEACONESS MEDICAL CENTER, INC. 2021-03-25 US claimed
US-20200129440-A1 COMPLEX FORMULATION COMPRISING HMG-COA REDUCTASE INHIBITOR AND CLOPIDOGREL DONG WHA PHARM. CO., LTD. (KR) 2020-04-30 US claimed
EP-2809319-B1 IMPROVEMENTS IN TEAR FILM STABILITY UNIV SYDNEY (AU) 2018-04-18 EP claimed
EP-2813509-B1 3,4,4a,10b-tetrahydro-1h-thiopyrano-[4,3-c]isoquinoline derivatives ASTRAZENECA AB (SE) 2017-02-01 EP claimed
EP-2521453-B1 COMBINATIONS OF VITAMIN D AND A STATIN FOR THE TREATMENT OF MIGRAINE HEADACHES BETH ISRAEL HOSPITAL (US) 2016-05-11 EP claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20150094447-A1 Novel Nitric Oxide Synthase Agonist Polymers PALMETTO PHARMACEUTICALS LLC (US) 2015-04-02 US claimed
US-8936635-B2 Bioresorbable nitric oxide agonist prodrug scaffolds for vascular stents PALMETTO PHARMACEUTICALS LLC (US) 2015-01-20 US claimed
EP-2813509-A1 3,4,4a,10b-tetrahydro-1h-thiopyrano-[4,3-c]isoquinoline derivatives Takeda GmbH (DE) 2014-12-17 EP claimed
EP-1505986-A1 COMBINATION OF AN HMG-CoA REDUCTASE INHIBITOR AND A NITRATE ESTER Scaramuzzino, Giovanni (IT) 2005-02-16 EP claimed
US-20040248972-A1 Compounds and uses thereof AMBIT BIOSCIENCES CORPORATION 2004-12-09 US claimed
WO-2004103960-A2 COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2004-12-02 WO claimed
US-20040053842-A1 Methods of treatment with CETP inhibitors and antihypertensive agents PFIZER INC. 2004-03-18 US claimed
US-20040048805-A1 Antilipemic agents SHIONOGI & CO., LTD. (JP) 2004-03-11 US claimed
US-20040039018-A1 CETP inhibitors in combination with antihypertensive agents and uses thereof PFIZER INC. 2004-02-26 US claimed
WO-2004004777-A1 USE OF CETP INHIBITORS AND ANTIHYPERTENSIVE AGENTS AS WELL AS OPTIONALLY HMG COA REDUCTASE INHIBITORS PFIZER PRODUCTS INC. (US) 2004-01-15 WO claimed
WO-2004004778-A1 USE OF CETP INHIBITORS AND OPTIONALLY HMG COA REDUCTABLE INHIBITORS AND/OR ANTIHYPERTENSIVE AGENTS PFIZER PRODUCTS INC. (US) 2004-01-15 WO claimed
WO-2003094923-A1 COMBINATION OF AN HMG-CoA REDUCTASE INHIBITOR AND A NITRATE ESTER SCARAMUZZINO GIOVANNI (IT) 2003-11-20 WO claimed
EP-1358879-A1 ANTILIPEMIC AGENTS SHIONOGI & CO., LTD. (JP) 2003-11-05 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040053842-A1 Methods of treatment with CETP inhibitors and antihypertensive agents CETP, APOB, MTTP HMGCR 9/4885
US-20040248972-A1 Compounds and uses thereof HMGCR, PCSK9, CYP46A1 HMGCR 1/4885
US-20040039018-A1 CETP inhibitors in combination with antihypertensive agents and uses thereof CETP, MTTP, APOB HMGCR 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.