SCHEMBL4952161

SCHEMBL4952161

C[C@]1(OC(=O)O)CSC(c2ccc(O)cc2O)=N1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 9/20 0.35
AMY1A P0DUB6 4/20 0.33
CSNK2A1 P68400 1/20 0.32
MAOB P27338 1/20 0.32
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA7 P43166 2/20 0.32
CA9 Q16790 2/20 0.32
CA14 Q9ULX7 2/20 0.32
PDK2 Q15119 1/20 0.32
PDK4 Q16654 1/20 0.32
ALDH1A1 P00352 2/20 0.32
ALOX5 P09917 1/20 0.32
TSHR P16473 1/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 2/20 0.32
ALOX12 P18054 2/20 0.32
HTT P42858 2/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28026304 0.91 TYR (0.36) TYRAMY1AMAOBCA12CA1
SCHEMBL6985974 0.87 KDM4E (0.37) AMY1ACSNK2A1CA12CA1CA2
SCHEMBL28067847 0.86 HSP90AB1 (0.35) TYRCA12CA1CA2CA7
SCHEMBL6987657 0.85 HTR2B (0.42) MAOBALDH1A1TSHRMAPTKDM4E
SCHEMBL28043436 0.83 TYR (0.35) TYRMAOBALDH1A1MAPTHTT
SCHEMBL6985038 0.82 HTR2B (0.36) ALDH1A1LMNAMAPTALOX12MEN1
SCHEMBL6986273 0.81 HTR2B (0.34) MAOBALDH1A1TSHRLMNAMAPT
Deferitrin SCHEMBL1272026 0.80 TYR (0.35) TYRAMY1AMAOBCA12CA1
Deferitrin SCHEMBL663744 0.80 TYR (0.35) TYRAMY1AMAOBCA12CA1
Deferitrin SCHEMBL18103545 0.80 TYR (0.35) TYRAMY1AMAOBCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1667727-B1 POLYAMINE-METAL CHELATOR CONJUGATES UNIV FLORIDA (US) 2008-07-09 EP claimed
EP-1302467-A2 Process for the preparation of substituted thiazoline derivatives and their intermediate DSM Fine Chemicals Austria Nfg GmbH & Co KG (AT) 2003-04-16 EP disclosed