SCHEMBL4953244

SCHEMBL4953244

Cc1ccc(-c2cnns2)c(-c2cnns2)[n+]1[O-]

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
GAA P10253 2/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 2/20 0.42
HTT P42858 2/20 0.42
RUNX1 Q01196 2/20 0.42
CBFB Q13951 2/20 0.42
GFER P55789 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4958231 0.73 ALDH1A1 (0.33) ALDH1A1GAAMAPTHPGDHTT
SCHEMBL4953247 0.72 ALDH1A1 (0.34) ALDH1A1GAAMAPTHPGDHTT
SCHEMBL4953518 0.70 ALDH1A1 (0.39) ALDH1A1GAAMAPTHPGDHTT
SCHEMBL4957173 0.68 ALDH1A1 (0.30) ALDH1A1GAAMAPTHPGDHTT
SCHEMBL4957177 0.62 ALDH1A1 (0.34) ALDH1A1GAAMAPTHPGDHTT
SCHEMBL6740529 0.60 ALDH1A1 (0.41) ALDH1A1GAAMAPTHPGDHTT
SCHEMBL6993258 0.57 ALDH1A1 (0.47) ALDH1A1GAAMAPTHPGDHTT
SCHEMBL10163319 0.56 METAP2 (0.41) ALDH1A1GAAMAPTHPGDHTT
SCHEMBL2345941 0.56
SCHEMBL6626713 0.55 GAA (0.41) ALDH1A1GAAMAPTHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed