SCHEMBL4958115

SCHEMBL4958115

COCCCN1CCOc2ccc(CO[C@H]3CN(C(=O)O)[C@H](CCOC)C[C@@H]3c3ccc(OC)cc3)cc21

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.35
THRB P10828 3/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
TP53 P04637 1/20 0.32
EDNRB P24530 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4646776 0.95 REN (0.34) RENTHRBCYP3A4CYP2C19ALDH1A1
SCHEMBL2925215 0.91 TP53 (0.37) RENTHRBALDH1A1TP53
SCHEMBL5503959 0.91 REN (0.36) RENTHRBCYP3A4CYP2C19ALDH1A1
SCHEMBL5507277 0.89 REN (0.36) RENTHRBCYP3A4CYP2C19ALDH1A1
SCHEMBL2922840 0.87 TMEM97 (0.35) RENALDH1A1TP53
SCHEMBL3945312 0.87 REN (0.32) RENEDNRB
SCHEMBL2917973 0.87 TMEM97 (0.35) RENALDH1A1TP53
SCHEMBL2923001 0.87 TMEM97 (0.35) RENALDH1A1TP53
SCHEMBL2921292 0.87 TMEM97 (0.35) RENALDH1A1TP53
SCHEMBL3945307 0.87 REN (0.33) RENTHRBCYP3A4CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1897879-A2 2,4,5 substituted piperidines as renin inhibitors Speedel Experimenta AG (CH) 2008-03-12 EP disclosed