SCHEMBL4646776

SCHEMBL4646776

COCCCN1CCOc2ccc(CO[C@H]3CN(C(=O)O)[C@H](CCC(=O)O)C[C@@H]3c3ccc(OC)cc3)cc21

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.34
THRB P10828 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2C19 P33261 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
PIK3CD O00329 1/20 0.31
PIK3CA P42336 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4958115 0.95 REN (0.35) RENTHRBCYP3A4CYP2C19ALDH1A1
SCHEMBL2917973 0.92 TMEM97 (0.35) RENALDH1A1
SCHEMBL5503959 0.89 REN (0.36) RENTHRBCYP3A4CYP2C19ALDH1A1
SCHEMBL5507277 0.88 REN (0.36) RENTHRBCYP3A4CYP2C19ALDH1A1
SCHEMBL3555798 0.87 ALDH1A1 (0.33) RENTHRBCYP3A4CYP2C19ALDH1A1
SCHEMBL2925215 0.87 TP53 (0.37) RENTHRBALDH1A1
SCHEMBL2923347 0.87 LMNA (0.36) ALDH1A1MAPTLMNA
SCHEMBL3903011 0.86 REN (0.36) REN
SCHEMBL2922840 0.86 TMEM97 (0.35) RENALDH1A1
SCHEMBL2917780 0.86 TP53 (0.34) RENALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1958634-A2 Substituted piperidines as inhibitors of beta-secretase, cathepsin D, plasmepsin II and/or HIV protease Speedel Experimenta AG (CH) 2008-08-20 EP disclosed