SCHEMBL4959867

SCHEMBL4959867

COCCN(C(=O)O)C1CCC(c2ccccc2)CNC1=O.[NaH]

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 6/20 0.36
LMNA P02545 3/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KDM4E B2RXH2 1/20 0.35
REN P00797 1/20 0.35
KCNH2 Q12809 1/20 0.35
SLC18A3 Q16572 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LIPE Q05469 1/20 0.35
ALDH1A1 P00352 2/20 0.34
ASAH1 Q13510 1/20 0.34
RAB9A P51151 1/20 0.34
MAPK1 P28482 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5559232 0.99 LMNA (0.36) NAAALMNAHTTNPSR1KDM4E
SCHEMBL5559237 0.99 LMNA (0.36) NAAALMNAHTTNPSR1KDM4E
SCHEMBL4959861 0.97 LMNA (0.35) NAAALMNAHTTNPSR1KDM4E
SCHEMBL5560000 0.81 CALCRL (0.38)
SCHEMBL5552436 0.74 HSD11B1 (0.37) NAAASLC18A3ALDH1A1ASAH1
SCHEMBL1197732 0.74 HSD11B1 (0.37) NAAASLC18A3ALDH1A1ASAH1
SCHEMBL1198609 0.74 HSD11B1 (0.37) NAAASLC18A3ALDH1A1ASAH1
SCHEMBL13225607 0.71 ABCB1 (0.35) NAAA
SCHEMBL15716250 0.70 CTSD (0.43) LMNARENKCNH2SMN1; SMN2MAPK1
SCHEMBL15716455 0.70 CTSD (0.43) LMNARENKCNH2SMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615914-A4 CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2008-03-12 EP disclosed
EP-1615914-A2 CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2006-01-18 EP disclosed
WO-2004091514-A2 CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2004-10-28 WO disclosed