SCHEMBL4960119

SCHEMBL4960119

COc1cc(C(COC(N)=O)n2ncnn2)cc(OC)c1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.34
MAPK1 P28482 1/20 0.34
PDK1 Q15118 1/20 0.34
TNF P01375 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
FKBP1A P62942 2/20 0.34
FKBP5 Q13451 2/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4959372 0.88 TNF (0.46) CYP17A1CYP2C9CYP2C19KDM4ELMNA
SCHEMBL4958557 0.81 TNF (0.44) CYP17A1CYP2C9CYP2C19KDM4ELMNA
SCHEMBL4957486 0.78 CYP1A2 (0.51) CYP2C19KDM4ELMNACYP1A2SMN1; SMN2
SCHEMBL4958071 0.76 CYP19A1 (0.51) CYP17A1CYP2C9CYP2C19CYP1A2SMN1; SMN2
SCHEMBL4959914 0.75 SLC6A2 (0.40) CYP17A1CYP2C9CYP2C19LMNACYP1A2
SCHEMBL4959908 0.75 ALDH1A1 (0.35) CYP17A1CYP2C9CYP2C19CYP1A2SMN1; SMN2
SCHEMBL4957281 0.75 SLC6A3 (0.56) CYP17A1CYP2C9CYP2C19LMNACYP1A2
SCHEMBL4959314 0.75 SLC6A2 (0.37) CYP17A1CYP2C9CYP2C19CYP1A2SMN1; SMN2
SCHEMBL4962094 0.75 SLC6A2 (0.32) CYP17A1CYP2C9CYP2C19CYP1A2SMN1; SMN2
SCHEMBL4958049 0.74 SLC6A2 (0.57) CYP17A1CYP2C9CYP2C19CYP1A2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879873-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK Holdings Co., Ltd. (KR) 2008-01-23 EP disclosed
WO-2006112685-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK HOLDINGS CO., LTD. (KR) 2006-10-26 WO disclosed