SCHEMBL4960580

SCHEMBL4960580

NC(=O)Nc1ccc2ncccc2c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.77
POLB P06746 2/20 0.77
MEN1 O00255 2/20 0.77
KMT2A Q03164 2/20 0.77
MAPT P10636 1/20 0.77
ALDH1A1 P00352 2/20 0.67
PABPC1 P11940 1/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
TSHR P16473 1/20 0.67
HSD17B10 Q99714 1/20 0.67
RAB9A P51151 7/20 0.62
CASP3 P42574 1/20 0.59
SENP8 Q96LD8 1/20 0.59
SENP7 Q9BQF6 1/20 0.59
SENP6 Q9GZR1 1/20 0.59
HTT P42858 2/20 0.58
NAMPT P43490 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
NOTUM Q6P988 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4972667 0.87 MEN1 (0.62) NPC1POLBMEN1KMT2AMAPT
SCHEMBL31054249 0.87 NPC1 (1.00) NPC1POLBMEN1KMT2AMAPT
SCHEMBL651929 0.87 NPC1 (1.00) NPC1POLBMEN1KMT2AMAPT
SCHEMBL30741445 0.85 NPC1 (0.79) NPC1POLBMEN1KMT2AMAPT
SCHEMBL4890353 0.85 NPC1 (0.79) NPC1POLBMEN1KMT2AMAPT
SCHEMBL28359062 0.85 ALDH1A1 (0.72) NPC1POLBMEN1KMT2AMAPT
SCHEMBL4526983 0.84 NPC1 (0.67) NPC1POLBMEN1KMT2AMAPT
SCHEMBL10310270 0.84 NPC1 (0.67) NPC1POLBMEN1KMT2AMAPT
SCHEMBL29944526 0.84 NPC1 (0.77) NPC1POLBMEN1KMT2AMAPT
SCHEMBL18885828 0.84 NPC1 (0.77) NPC1POLBMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630373-A1 INDOLE DERIVATIVES AS 5HT1C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-12-28 EP claimed
CN-108658869-A Compound with anti-tumor activity and preparation method thereof and the purposes in pharmacy 复旦大学 2018-10-16 CN disclosed
EP-1969051-A2 INHIBITORS OF FATTY ACID AMIDE HYDROLASE N.V. Organon (NL) 2008-09-17 EP disclosed
WO-2008024139-A2 INHIBITORS OF FATTY ACID AMIDE HYDROLASE N.V. ORGANON (NL) 2008-02-28 WO disclosed
WO-2007079180-A2 INHIBITORS OF FATTY ACID AMIDE HYDROLASE N.V. ORGANON (NL) 2007-07-12 WO disclosed