SCHEMBL4960652

SCHEMBL4960652

O=C(O)c1cccn1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
APEX1 P27695 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SRD5A2 P31213 2/20 0.44
AHSA1 O95433 1/20 0.43
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
NOTUM Q6P988 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CA12 O43570 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
RECQL P46063 1/20 0.38
KIF11 P52732 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6052408 0.82 TDP1 (0.50) POLBAPEX1TDP1L3MBTL1AHSA1
SCHEMBL29006050 0.82 AHSA1 (0.40) AHSA1CES2CES1NOTUMCA12
SCHEMBL4543597 0.82 POLB (0.41) POLBAPEX1TDP1L3MBTL1AHSA1
SCHEMBL4787559 0.81 POLB (0.61) POLBAPEX1TDP1L3MBTL1NOTUM
SCHEMBL26601277 0.79 KDM4E (0.47) POLBAPEX1TDP1L3MBTL1SRD5A2
SCHEMBL20917138 0.79 POLB (0.50) POLBAPEX1TDP1L3MBTL1NPC1
SCHEMBL15058294 0.79 POLB (0.50) POLBAPEX1TDP1L3MBTL1NOTUM
SCHEMBL7630480 0.79 RECQL (0.57) POLBAPEX1TDP1L3MBTL1NOTUM
SCHEMBL4540045 0.79 L3MBTL1 (0.50) POLBAPEX1TDP1L3MBTL1ALDH1A1
SCHEMBL29797734 0.79 POLB (0.41) POLBAPEX1TDP1L3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1044364-B8 METHOD FOR THE QUANTIFICATION OF SOLID-PHASE REACTIONS USING FLUORINE NMR AVENTIS PHARMA INC (US) 2008-01-02 EP disclosed
EP-1044364-B1 METHOD FOR THE QUANTIFICATION OF SOLID-PHASE REACTIONS USING FLUORINE NMR AVENTIS PHARM PROD INC (US) 2007-06-13 EP disclosed
EP-1044364-A4 METHOD AND REAGENTS FOR THE QUANTIFICATION OF SOLID-PHASE REACTIONS USING FLUORINE NMR AVENTIS PHARM PROD INC (US) 2004-10-06 EP disclosed
US-6599753-B1 Quantifying a solid-phase reaction; obtain chemical intermediate, incubate with fluorine compound, expose to nuclear magnetic resonance, monitor intensity, compare to control AVENTIS PHARMACEUTICALS INC. 2003-07-29 US disclosed
EP-1044364-A1 METHOD AND REAGENTS FOR THE QUANTIFICATION OF SOLID-PHASE REACTIONS USING FLUORINE NMR Aventis Pharmaceuticals Products Inc. (US) 2000-10-18 EP disclosed
WO-1999031491-A1 METHOD AND REAGENTS FOR THE QUANTIFICATION OF SOLID-PHASE REACTIONS USING FLUORINE NMR AVENTIS PHARMACEUTICALS PRODUCTS INC. (US) 1999-06-24 WO disclosed