SCHEMBL4963643

SCHEMBL4963643

CCC(O)Cc1csc(NS(=O)(=O)c2ccc(OCCCN3CCOCC3)cc2C)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.42
UBE2N P61088 1/20 0.41
TRPV4 Q9HBA0 1/20 0.40
MCL1 Q07820 1/20 0.40
HRH3 Q9Y5N1 3/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 2/20 0.40
CYP1A2 P05177 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
HTR2A P28223 1/20 0.40
SCN1A P35498 1/20 0.40
HTR2B P41595 1/20 0.40
KCNH2 Q12809 1/20 0.40
SCN2A Q99250 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
SCN3A Q9NY46 1/20 0.40
EPHX2 P34913 4/20 0.40
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4964680 0.96 MEN1 (0.43) ROCK1UBE2NTRPV4ALDH1A1MEN1
SCHEMBL4969260 0.92 ROCK1 (0.42) ROCK1UBE2NTRPV4MCL1HRH3
SCHEMBL4964132 0.86 ROCK1 (0.42) ROCK1UBE2NTRPV4MCL1HRH3
SCHEMBL4968167 0.83 ROCK1 (0.41) ROCK1UBE2NTRPV4MCL1HRH3
SCHEMBL4969661 0.83 HSD11B1 (0.44) ROCK1TRPV4MCL1HRH3ALDH1A1
SCHEMBL4965583 0.82 NPC1 (0.43) ROCK1UBE2NTRPV4ALDH1A1MEN1
SCHEMBL4963884 0.82 ROCK1 (0.40) ROCK1UBE2NTRPV4MCL1HRH3
SCHEMBL4962659 0.82 HRH3 (0.42) ROCK1UBE2NHRH3SIGMAR1EPHX2
SCHEMBL4964526 0.81 HRH3 (0.43) ROCK1UBE2NHRH3SIGMAR1EPHX2
SCHEMBL4968708 0.81 HSD11B1 (0.41) TRPV4ALDH1A1SCN1AEPHX2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed