SCHEMBL4965583

SCHEMBL4965583

CCC(O)(CC)Cc1csc(NS(=O)(=O)c2ccc(OCCN3CCOCC3)cc2C)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
ROCK1 Q13464 2/20 0.41
MMP1 P03956 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
GAA P10253 1/20 0.38
UBE2N P61088 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
ULK1 O75385 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4964132 0.96 ROCK1 (0.42) NPC1SMN1; SMN2ALDH1A1ROCK1UBE2N
SCHEMBL4966824 0.92 NPC1 (0.42) NPC1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL4964680 0.86 MEN1 (0.43) NPC1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL4963210 0.85 TRPV4 (0.40) MEN1KMT2ASMN1; SMN2KDM4EALDH1A1
SCHEMBL4966468 0.84 TRPV4 (0.39) MEN1KMT2ASMN1; SMN2KDM4EALDH1A1
SCHEMBL4966984 0.84 HDAC3 (0.48) SMN1; SMN2ALDH1A1ROCK1CA12CA1
SCHEMBL4970500 0.83 HSD11B1 (0.44) NPC1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL4964824 0.83 EPHX2 (0.49) SMN1; SMN2KDM4EALDH1A1ROCK1TRPV4
SCHEMBL4966262 0.83 KMT2A (0.40) MEN1KMT2AKDM4EALDH1A1HSD11B1
SCHEMBL4963643 0.82 ROCK1 (0.42) NPC1MEN1KMT2AALDH1A1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed