SCHEMBL4964175

SCHEMBL4964175

O=C1Cc2c(cc(Cc3cccc(F)c3)cc2C2CCNCC2)N1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.44
SLC6A2 P23975 8/20 0.39
SLC6A3 Q01959 8/20 0.39
SLC6A4 P31645 6/20 0.39
HTR1A P08908 4/20 0.39
PLG P00747 1/20 0.36
DAO P14920 1/20 0.35
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
CCR2 P41597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4962936 0.99 HTR6 (0.43) HTR6SLC6A2SLC6A3SLC6A4HTR1A
SCHEMBL4967691 0.94 HTR6 (0.39) HTR6SLC6A2SLC6A3SLC6A4HTR1A
SCHEMBL4965972 0.82 HTR6 (0.44) HTR6SLC6A2SLC6A3SLC6A4HTR1A
SCHEMBL4977286 0.76 HTR6 (0.38) HTR6SLC6A2SLC6A3SLC6A4HTR1A
SCHEMBL152514 0.73 HTR2C (0.45) HTR6SLC6A2SLC6A3SLC6A4HTR1A
SCHEMBL4962966 0.72 DRD2 (0.48)
SCHEMBL3854328 0.67 KMT2A (0.47) HTR6SLC6A2SLC6A3SLC6A4HTR1A
Hydrochloric Acid SCHEMBL3856321 0.67 KMT2A (0.47) HTR6SLC6A2SLC6A3SLC6A4HTR1A
SCHEMBL14597077 0.65 HTR6 (0.46) HTR6SLC6A2SLC6A3SLC6A4HTR1A
SCHEMBL17974655 0.64 PDK2 (0.44) HTR1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904483-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. Hoffmann-Roche AG (CH) 2008-04-02 EP claimed
WO-2007006677-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO claimed
EP-1904483-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. Hoffmann-Roche AG (CH) 2008-04-02 EP disclosed
WO-2007006677-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed