SCHEMBL4977286

SCHEMBL4977286

O=C1[N]c2c(cc(Cc3cccc(F)c3)cc2C2CCNC2)N1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.38
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
HTR2A P28223 1/20 0.36
SLC6A2 P23975 4/20 0.35
SLC6A3 Q01959 4/20 0.35
CCR2 P41597 1/20 0.35
PLG P00747 1/20 0.34
SLC6A4 P31645 2/20 0.33
CDK9 P50750 1/20 0.33
DAO P14920 1/20 0.33
HTR1A P08908 1/20 0.33
MPO P05164 1/20 0.33
ADRA1A P35348 1/20 0.32
HRH1 P35367 1/20 0.32
ADRA1B P35368 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4965972 0.94 HTR6 (0.44) HTR6HTR2CHTR2BSLC6A2SLC6A3
SCHEMBL4966050 0.88 GABRA1 (0.38) SLC6A2SLC6A3SLC6A4HTR1AHRH1
Hydrochloric Acid SCHEMBL4966442 0.87 GABRA1 (0.38) SLC6A2SLC6A3SLC6A4HTR1AHRH1
SCHEMBL4977909 0.84 CXCR2 (0.34) SLC6A2SLC6A3SLC6A4HTR1AMPO
SCHEMBL4967691 0.82 HTR6 (0.39) HTR6HTR2CHTR2BHTR2ASLC6A2
SCHEMBL4964175 0.76 HTR6 (0.44) HTR6HTR2CHTR2BSLC6A2SLC6A3
Hydrochloric Acid SCHEMBL4962936 0.75 HTR6 (0.43) HTR6HTR2CHTR2BSLC6A2SLC6A3
SCHEMBL4965409 0.72 GABRA1 (0.40) HTR2CHTR2BHTR2ASLC6A2SLC6A3
SCHEMBL4964731 0.69 KIT (0.42) SLC6A2SLC6A3SLC6A4HRH1
SCHEMBL4964772 0.68 HRH1 (0.51) HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904483-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. Hoffmann-Roche AG (CH) 2008-04-02 EP claimed
WO-2007006677-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO claimed