SCHEMBL4965181

SCHEMBL4965181

O=C(Nc1ccc(Cl)c(NC(=O)c2ccc(Cl)cc2)c1)c1cccnc1

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.71
RAB9A P51151 4/20 0.70
NPC1 O15118 3/20 0.70
L3MBTL1 Q9Y468 2/20 0.66
NAMPT P43490 1/20 0.64
CYP11B1 P15538 1/20 0.64
CYP11B2 P19099 1/20 0.64
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
ALDH1A1 P00352 4/20 0.60
KCNMA1 Q12791 1/20 0.60
KDM4E B2RXH2 1/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
MAPT P10636 3/20 0.60
HTT P42858 1/20 0.60
KCNK3 O14649 1/20 0.59
LMNA P02545 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5897778 0.88 TSHR (0.65) TSHRRAB9ANPC1L3MBTL1CYP11B1
SCHEMBL403822 0.87 TSHR (0.67) TSHRRAB9ANPC1L3MBTL1MEN1
SCHEMBL11090153 0.84 NAMPT (0.78) RAB9ANPC1L3MBTL1NAMPTCYP11B1
SCHEMBL398150 0.84 TSHR (0.66) TSHRRAB9ANPC1L3MBTL1NAMPT
SCHEMBL27903120 0.83 RAB9A (1.00) TSHRRAB9ANPC1L3MBTL1MEN1
SCHEMBL403003 0.82 KCNQ3 (0.68) RAB9AMEN1KMT2AALDH1A1KDM4E
SCHEMBL15683903 0.81 TSHR (0.57) TSHRRAB9ANPC1L3MBTL1MEN1
SCHEMBL15683400 0.80 ALDH1A1 (0.56) TSHRRAB9ANPC1L3MBTL1MEN1
SCHEMBL3790049 0.80 MAPT (0.83) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL14426548 0.80 RAB9A (0.78) TSHRRAB9ANPC1L3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957461-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING Genentech, Inc. (US) 2008-08-20 EP disclosed
WO-2007059157-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING GENENTECH, INC. (US) 2007-05-24 WO disclosed