SCHEMBL4965573

SCHEMBL4965573

Cc1cc(Br)ccc1S(=O)(=O)Nc1nc(CC2(O)CCC2)cs1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
POLB P06746 2/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
ALDH1A1 P00352 3/20 0.38
HSD11B1 P28845 3/20 0.37
HSD17B1 P14061 2/20 0.37
HSD17B2 P37059 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM1A O60341 2/20 0.36
MAOA P21397 2/20 0.36
PKM P14618 1/20 0.35
BRD4 O60885 1/20 0.35
BRD1 O95696 1/20 0.35
BRPF1 P55201 1/20 0.35
BRPF3 Q9ULD4 1/20 0.35
GHSR Q92847 1/20 0.35
SCN5A Q14524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3608648 0.80 KMT2A (0.49) KMT2AMEN1POLBALDH1A1HSD11B1
SCHEMBL4963075 0.78 HSD11B1 (0.61) KMT2AMEN1POLBALDH1A1HSD11B1
SCHEMBL4963016 0.76 HSD11B1 (0.61) KMT2AMEN1POLBALDH1A1HSD11B1
SCHEMBL3625053 0.74 HSD11B1 (0.61) KMT2AMEN1POLBALDH1A1HSD11B1
SCHEMBL4968167 0.74 ROCK1 (0.41) ALDH1A1
SCHEMBL4964152 0.73 CA1 (0.40) KMT2AMEN1POLBCA1CA2
SCHEMBL4967012 0.70 HSD11B1 (0.58) KMT2AMEN1POLBHSD11B1HSD17B1
SCHEMBL7140715 0.69 KMT2A (0.46) KMT2AMEN1POLBALDH1A1HSD11B1
SCHEMBL27650013 0.69 KMT2A (0.63) KMT2AMEN1POLBALDH1A1CYP2C9
SCHEMBL3622234 0.68 KMT2A (0.45) KMT2AMEN1POLBALDH1A1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed