SCHEMBL4964152

SCHEMBL4964152

CCC(O)(CC)c1csc(NS(=O)(=O)c2ccc(Br)cc2C)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
KDM1A O60341 3/20 0.39
MAOA P21397 2/20 0.39
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
MAPK1 P28482 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
POLB P06746 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
HSD17B1 P14061 1/20 0.37
HSD11B1 P28845 1/20 0.37
HSD17B2 P37059 1/20 0.37
ALDH1A1 P00352 3/20 0.37
BRD4 O60885 1/20 0.37
BRD1 O95696 1/20 0.37
BRPF1 P55201 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4966328 0.88 CA1 (0.44) CA1CA2KDM1AMAOAKMT2A
SCHEMBL4964537 0.86 MEN1 (0.43) KDM1AMAOAKMT2AMEN1MAPK1
SCHEMBL4964673 0.83 KDM1A (0.53) KDM1AMAOAKMT2AMEN1HSD17B2
SCHEMBL4963943 0.82 KDM4E (0.47) KDM1AMAOAMAPK1SMN1; SMN2KDM4E
SCHEMBL4965545 0.80 KMT2A (0.46) KDM1AMAOAKMT2AMEN1SMN1; SMN2
SCHEMBL4964519 0.78 NPSR1 (0.42) KDM1AMAOAKMT2AMEN1SMN1; SMN2
SCHEMBL4965534 0.77 SMN1; SMN2 (0.53) KDM1AMAOAKMT2AMEN1SMN1; SMN2
SCHEMBL4965845 0.77 HSD11B1 (0.61) KDM1AMAOAKMT2AMEN1POLB
SCHEMBL3608648 0.77 KMT2A (0.49) KMT2AMEN1POLBGAAMAPT
SCHEMBL4969440 0.76 HCRTR1 (0.47) KDM1AMAOAKMT2AMEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed