SCHEMBL4965859

SCHEMBL4965859

O=C(O)c1c[nH]c(=O)c(C2CCCC(c3ccccc3)C2)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.43
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C1 Q04828 1/20 0.39
TRPV6 Q9H1D0 1/20 0.37
CYP2D6 P10635 1/20 0.36
P2RY14 Q15391 1/20 0.36
RARG P13631 2/20 0.36
RARB P10826 1/20 0.36
LIPG Q9Y5X9 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967987 0.95 AKR1C3 (0.44) KMOALDH1A1KDM4EMEN1GAA
SCHEMBL4969223 0.82 NOTUM (0.43) KMO
SCHEMBL4969319 0.82 NOTUM (0.39) KMOALDH1A1MEN1KMT2ARARG
SCHEMBL4966863 0.81 RAB9A (0.45) KMOKDM4EMEN1KMT2A
SCHEMBL6209027 0.79 NOTUM (0.46) KMOALDH1A1KDM4EMEN1GAA
Bicarbonate SCHEMBL7568966 0.73 AKR1C3 (0.60) KMOAKR1C3AKR1C1
SCHEMBL9471737 0.70 CYP2D6 (0.50) KMOALDH1A1KDM4EKMT2AAKR1C3
SCHEMBL780234 0.70 AKR1C3 (0.52) AKR1C3AKR1C1
SCHEMBL7568960 0.68 AKR1C3 (0.58) KMOAKR1C3AKR1C1
Bicarbonate SCHEMBL11121465 0.66 AKR1C3 (0.53) KMOAKR1C3AKR1C1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954693-A1 BETA-SECRETASE MODULATORS AND METHODS OF USE Amgen Inc. (US) 2008-08-13 EP disclosed
WO-2007062007-A1 BETA-SECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2007-05-31 WO disclosed