SCHEMBL4966498

SCHEMBL4966498

O=Cc1cc(-c2ccccc2I)c(F)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.37
ERN1 O75460 3/20 0.33
C1R P00736 3/20 0.33
MCL1 Q07820 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
LMNA P02545 2/20 0.32
THRB P10828 1/20 0.32
BLM P54132 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HTT P42858 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
PTGS2 P35354 2/20 0.30
KCNN4 O15554 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18133931 0.74 TDP1 (0.43) TDP1ERN1MCL1ALDH1A1
SCHEMBL1053001 0.73 TDP1 (0.50) TDP1ERN1MEN1KMT2ALMNA
SCHEMBL24028007 0.72 ALDH1A1 (0.39) TDP1ERN1MEN1KMT2AALDH1A1
SCHEMBL24500913 0.72 LMNA (0.52) TDP1ERN1MCL1MEN1KMT2A
SCHEMBL4844978 0.70 ERN1 (0.46) TDP1ERN1MEN1KMT2ALMNA
SCHEMBL27196550 0.70 ERN1 (0.37) TDP1ERN1
SCHEMBL6187165 0.69 TDP1 (0.46) TDP1ERN1MEN1KMT2ALMNA
SCHEMBL11387443 0.69 MEN1 (0.46) TDP1MCL1MEN1KMT2ALMNA
SCHEMBL30525125 0.68 TDP1 (0.33) TDP1ERN1ALDH1A1
SCHEMBL29055095 0.68 TDP1 (0.33) TDP1ERN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881990-A1 PROCESSES FOR PREPARING OF GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZENE DERIVATIVES AND INTERMEDIATES THEREIN Boehringer Ingelheim International GmbH (DE) 2008-01-30 EP disclosed
WO-2006120208-A1 PROCESSES FOR PREPARING OF GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZENE DERIVATIVES AND INTERMEDIATES THEREIN BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-11-16 WO disclosed