SCHEMBL4967758

SCHEMBL4967758

COc1ccc(Cc2cc(Br)c(SC)cc2N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.41
LTA4H P09960 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP2D6 P10635 1/20 0.41
ATM Q13315 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
CASP3 P42574 1/20 0.40
RAB9A P51151 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
HTR2A P28223 1/20 0.39
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.38
IDO1 P14902 2/20 0.38
AGXT P21549 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4966913 0.85 NPC1 (0.36) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL4969623 0.84 HTR2A (0.49) MPOLTA4HALDH1A1CYP2D6ATM
SCHEMBL4967204 0.81 MAOB (0.45) LTA4HALDH1A1MEN1KMT2AHTR2A
SCHEMBL4968294 0.81 HTR2A (0.39) MPOLTA4HALDH1A1CYP2D6ATM
SCHEMBL4967818 0.79 DHFR (0.40) MPOLTA4HALDH1A1CYP2D6ATM
SCHEMBL4967755 0.77 MAPT (0.44) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL6160744 0.76 LTA4H (0.50) MPOLTA4HALDH1A1CYP2D6ATM
SCHEMBL4967785 0.75 PDE4A (0.41) MPOALDH1A1MEN1KMT2AHTR2A
SCHEMBL12110695 0.73 TDP1 (0.50) MPOLTA4HALDH1A1CYP2D6ATM
SCHEMBL3902050 0.73 LTA4H (0.60) LTA4HALDH1A1CYP2D6ATMMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed