SCHEMBL4968294

SCHEMBL4968294

COc1ccc(Cc2cc(Br)c(OC(C)C)cc2N)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.39
SLC6A4 P31645 1/20 0.39
MPO P05164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP2D6 P10635 1/20 0.38
ATM Q13315 1/20 0.38
LMNA P02545 1/20 0.37
LTA4H P09960 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4969623 0.88 HTR2A (0.49) HTR2AMPOALDH1A1CYP2D6ATM
SCHEMBL4966698 0.86 CSNK2A1 (0.36) HTR2ASMN1; SMN2ALDH1A1
SCHEMBL4967818 0.83 DHFR (0.40) HTR2AMPOSMN1; SMN2ALDH1A1CYP2D6
SCHEMBL4969232 0.81 MAOB (0.40) HTR2ASLC6A4ALDH1A1CYP2D6LMNA
SCHEMBL4967758 0.81 MPO (0.41) HTR2AMPOALDH1A1CYP2D6ATM
SCHEMBL4967785 0.79 PDE4A (0.41) HTR2ASLC6A4MPOALDH1A1LMNA
SCHEMBL4965832 0.77 FPR1 (0.42) SMN1; SMN2ALDH1A1LMNA
SCHEMBL1252319 0.76 ALDH1A1 (0.44) HTR2ASMN1; SMN2ALDH1A1
SCHEMBL4971131 0.73 PDE4D (0.40)
SCHEMBL14116480 0.73 PDE4D (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed