SCHEMBL4968684

SCHEMBL4968684

CC(=O)N1CCN(c2ccc(C(=O)Nc3ccc(Cl)c(Nc4ccc(F)cc4)c3)c(C)n2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
USP2 O75604 1/20 0.44
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
NPY1R P25929 1/20 0.44
NPY2R P49146 1/20 0.44
MT-CO2 P00403 1/20 0.43
LMNA P02545 3/20 0.42
MAPT P10636 2/20 0.42
TRPV1 Q8NER1 1/20 0.42
IKBKB O14920 1/20 0.42
BPTF Q12830 1/20 0.42
EGFR P00533 1/20 0.41
CTNNB1 P35222 1/20 0.40
TCF7L2 Q9NQB0 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL400967 0.91 NPC1 (0.46) ALDH1A1USP2TP53HPGDMAPK1
SCHEMBL4970783 0.88 KMT2A (0.47) ALDH1A1USP2TP53HPGDMAPK1
SCHEMBL4970534 0.83 SMO (0.50) NPY1RNPY2RTRPV1IKBKB
SCHEMBL4971048 0.83 RAB9A (0.50) ALDH1A1MAPK1LMNAMAPTEGFR
SCHEMBL403228 0.82 NPC1 (0.58) ALDH1A1USP2TP53HPGDMAPK1
SCHEMBL4977786 0.81 NPY1R (0.54) NPY1RNPY2RMAPTTRPV1
SCHEMBL401245 0.79 NPC1 (0.46) ALDH1A1HPGDNPY1RNPY2RMAPT
SCHEMBL1068026 0.77 ALB (0.54) ALDH1A1USP2TP53HPGDMAPK1
SCHEMBL4975360 0.77 CYP2C9 (0.56)
SCHEMBL4971825 0.76 RAB9A (0.54) ALDH1A1HPGDMAPK1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957461-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING Genentech, Inc. (US) 2008-08-20 EP disclosed
WO-2007059157-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING GENENTECH, INC. (US) 2007-05-24 WO disclosed