SCHEMBL4968929

SCHEMBL4968929

Clc1ccc2cccc(N3CCNCC3)c2n1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.63
HTR2C P28335 2/20 0.63
SLC6A4 P31645 1/20 0.63
HTR3E A5X5Y0 2/20 0.55
HTR3B O95264 2/20 0.55
HTR3A P46098 2/20 0.55
HTR3D Q70Z44 2/20 0.55
HTR3C Q8WXA8 2/20 0.55
ALDH1A1 P00352 2/20 0.55
ADRB1 P08588 3/20 0.53
HTR6 P50406 4/20 0.53
DRD2 P14416 3/20 0.53
HTR1A P08908 3/20 0.53
HTR5A P47898 2/20 0.53
DRD3 P35462 2/20 0.53
HTR7 P34969 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
NCF1 P14598 1/20 0.53
TSHR P16473 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3560188 0.81 HTR2A (0.63) HTR2AHTR2CSLC6A4HTR3EHTR3B
Hydrochloric Acid SCHEMBL4008999 0.80 HTR2A (0.61) HTR2AHTR2CSLC6A4HTR3EHTR3B
SCHEMBL5379037 0.78 HTR2A (0.58) HTR2AHTR2CSLC6A4HTR3EHTR3B
SCHEMBL5223620 0.78 HTR2A (0.58) HTR2AHTR2CSLC6A4HTR3EHTR3B
SCHEMBL5373371 0.78 HTR2A (0.58) HTR2AHTR2CSLC6A4HTR3EHTR3B
SCHEMBL4014210 0.78 HTR2A (0.58) HTR2AHTR2CSLC6A4HTR3EHTR3B
SCHEMBL1045944 0.78 HTR2A (1.00) HTR2AHTR2CSLC6A4HTR3EHTR3B
Hydrochloric Acid SCHEMBL1048620 0.76 HTR2A (0.97) HTR2AHTR2CSLC6A4HTR3EHTR3B
SCHEMBL3560924 0.75 HTR6 (0.56) HTR2AHTR2CSLC6A4HTR3EHTR3B
SCHEMBL5372201 0.75 HTR2A (0.58) HTR2AHTR2CSLC6A4HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888559-A2 PIPERAZINE-PIPERIDINE ANTAGONISTS AND AGONISTS OF THE 5-HT1A RECEPTOR Wyeth a Corporation of the State of Delaware (US) 2008-02-20 EP disclosed
WO-2006135839-A2 PIPERAZINE-PIPERIDINE ANTAGONISTS AND AGONISTS OF THE 5-HT1A RECEPTOR WYETH (US) 2006-12-21 WO disclosed