Benzimidazole

Benzimidazole

SCHEMBL4969244

O=P(O)(O)O.O=P(O)(O)O.O=P(O)(O)O.c1ccc2[nH]cnc2c1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Benzimidazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
RAB9A P51151 3/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
HTT P42858 1/20 0.47
PARP1 P09874 2/20 0.46
PDPK1 O15530 1/20 0.46
CA12 O43570 1/20 0.46
ALOX15 P16050 1/20 0.46
CA9 Q16790 1/20 0.46
TNKS2 Q9H2K2 1/20 0.46
HDAC6 Q9UBN7 1/20 0.45
CTNNB1 P35222 1/20 0.44
WNT3A P56704 1/20 0.44
QPCT Q16769 1/20 0.44
QPCTL Q9NXS2 1/20 0.44
POLB P06746 2/20 0.41
CASP6 P55212 2/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzimidazole SCHEMBL1760296 1.00 SMN1; SMN2 (0.47) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Benzimidazole SCHEMBL31595948 1.00 SMN1; SMN2 (0.47) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Benzimidazole SCHEMBL15092883 0.92 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Benzimidazole SCHEMBL28459336 0.92 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Benzimidazole SCHEMBL28471251 0.92 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Benzimidazole SCHEMBL28467053 0.92 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Benzimidazole SCHEMBL7068655 0.92 SMN1; SMN2 (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Benzimidazole SCHEMBL28462564 0.92 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Pyrophosphoric Acid SCHEMBL28258905 0.89 SMN1; SMN2 (0.43) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD
Benzimidazole SCHEMBL28459334 0.88 SMN1; SMN2 (0.46) SMN1; SMN2RAB9AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1777300-B1 Organic salt additives for nucleic acid amplification ROCHE DIAGNOSTICS GMBH (DE) 2008-08-27 EP disclosed