SCHEMBL4969440

SCHEMBL4969440

CCC(O)(CC)c1csc(NS(=O)(=O)c2cccc3ccccc23)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.47
CCR4 P51679 1/20 0.45
MAPT P10636 1/20 0.45
RORA P35398 1/20 0.45
RORC P51449 1/20 0.45
NR1H2 P55055 1/20 0.45
NR1H4 Q96RI1 1/20 0.45
EDNRB P24530 2/20 0.43
EDNRA P25101 2/20 0.43
KCNA5 P22460 1/20 0.43
TSHR P16473 1/20 0.43
ALDH1A1 P00352 3/20 0.42
PKM P14618 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
USP2 O75604 1/20 0.42
USP8 P40818 1/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B1 P14061 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4965815 0.86 PDPK1 (0.48) CCR4ALDH1A1PKMMAPK1SMN1; SMN2
SCHEMBL4963934 0.83 HSD11B1 (0.49) CCR4HSD17B1HSD11B1HSD17B2KDM1A
SCHEMBL4965845 0.82 HSD11B1 (0.61) CCR4EDNRBEDNRAHSD17B1HSD11B1
SCHEMBL4962685 0.81 MEN1 (0.60) MAPTALDH1A1PKMSMN1; SMN2CYP2C9
SCHEMBL4963696 0.79 CCR2 (0.43) ALDH1A1PKMCYP2C9CYP2C19MEN1
SCHEMBL4963943 0.78 KDM4E (0.47) CCR4EDNRBEDNRATSHRALDH1A1
SCHEMBL4965824 0.78 KMT2A (0.51) MAPTALDH1A1PKMCYP2C9CYP2C19
SCHEMBL4964568 0.78 CCR2 (0.45) MAPTSMN1; SMN2
SCHEMBL4966790 0.78 KDM1A (0.45) ALDH1A1CYP2C9CYP2C19MEN1KMT2A
SCHEMBL4965561 0.77 KMT2A (0.54) ALDH1A1PKMSMN1; SMN2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed