SCHEMBL4969587

SCHEMBL4969587

NC(Cc1ccccc1)C(=O)N1CCC(NC(=O)c2ccccc2)C1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 5/20 0.61
POLB P06746 1/20 0.53
OPRD1 P41143 1/20 0.52
ROCK2 O75116 1/20 0.52
CYP3A4 P08684 1/20 0.52
HDAC8 Q9BY41 2/20 0.51
DRD2 P14416 1/20 0.51
DRD4 P21917 1/20 0.51
NPSR1 Q6W5P4 1/20 0.50
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
CTSK P43235 1/20 0.50
KDM5A P29375 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6705226 0.85 HDAC8 (0.56) SMYD3POLBOPRD1ROCK2CYP3A4
Hydrochloric Acid SCHEMBL4883454 0.85 MCHR1 (0.64) SMYD3POLBDRD2DRD4
Hydrochloric Acid SCHEMBL4602478 0.85 MCHR1 (0.64) SMYD3POLBDRD2DRD4
SCHEMBL6164884 0.82 OPRD1 (0.60) SMYD3POLBOPRD1ROCK2CYP3A4
SCHEMBL2400255 0.81 DPP4 (0.57) SMYD3
SCHEMBL2400261 0.81 DPP4 (0.57) SMYD3
SCHEMBL26814547 0.80 NPSR1 (0.60) POLBNPSR1CTSLCTSBCTSK
SCHEMBL4086820 0.79 HDAC8 (0.59) POLBOPRD1HDAC8
SCHEMBL4095232 0.79 HDAC8 (0.59) POLBOPRD1HDAC8
SCHEMBL6052747 0.79 HDAC8 (0.59) POLBOPRD1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966130-A2 MODIFIED LYSINE-MIMETIC COMPOUNDS Zealand Pharma A/S (DK) 2008-09-10 EP claimed
WO-2007078990-A2 MODIFIED LYSINE-MIMETIC COMPOUNDS ZEALAND PHARMA A/S (DK) 2007-07-12 WO claimed