SCHEMBL4969713

SCHEMBL4969713

O=C(Cc1ccccc1)c1ccc(Br)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
SRD5A2 P31213 2/20 0.50
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
PLAU P00749 1/20 0.50
KDM4E B2RXH2 1/20 0.50
NPC1 O15118 1/20 0.50
GAA P10253 2/20 0.45
ALDH1A1 P00352 4/20 0.44
POLB P06746 1/20 0.44
GRM1 Q13255 1/20 0.44
STS P08842 1/20 0.43
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27955217 0.87 MAPT (0.56) MAPTL3MBTL1SRD5A2RAB9ASMN1; SMN2
SCHEMBL1515798 0.85 MAPT (0.61) MAPTL3MBTL1SRD5A2RAB9ASMN1; SMN2
SCHEMBL15100944 0.81 MAPT (0.60) MAPTL3MBTL1SRD5A2RAB9ASMN1; SMN2
SCHEMBL1515782 0.81 MAPT (0.60) MAPTL3MBTL1SRD5A2RAB9ASMN1; SMN2
SCHEMBL4846480 0.80 MAPT (0.53) MAPTL3MBTL1SRD5A2RAB9ASMN1; SMN2
SCHEMBL14533992 0.79 MAPT (0.57) MAPTL3MBTL1SRD5A2RAB9ASMN1; SMN2
SCHEMBL4949504 0.78 ACHE (0.42) MAPTRAB9ANPC1ALDH1A1POLB
SCHEMBL2953875 0.78 PTPN1 (0.57) CES2CES1
SCHEMBL1515818 0.77 L3MBTL1 (0.65) MAPTL3MBTL1SRD5A2RAB9ASMN1; SMN2
SCHEMBL3497492 0.77 KMT2A (0.58) MAPTL3MBTL1RAB9ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008099020-A1 1,1-DIOXO-1-THIA-5,10-DIAZADIBENZOCYCLOHEPTENES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed
WO-2008099020-A1 1,1-DIOXO-1-THIA-5,10-DIAZADIBENZOCYCLOHEPTENES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed