SCHEMBL4970728

SCHEMBL4970728

CC1(C)CC(CC=O)Nc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.40
ADRA2A P08913 4/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 2/20 0.37
AKR1B1 P15121 2/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967797 0.81 CA9 (0.34) MAPTKMT2AMEN1GAA
SCHEMBL4017459 0.78 PNMT (0.42) PNMTADRA2AADRA2BADRA2C
SCHEMBL6187691 0.78 AKR1B1 (0.39) PNMTADRA2AADRA2BADRA2CMAPT
SCHEMBL28101785 0.70 AKR1B1 (0.41) PNMTADRA2AADRA2BADRA2CMAPT
SCHEMBL2061536 0.70 AKR1B1 (0.44) PNMTADRA2AADRA2BADRA2CMAPT
SCHEMBL2062098 0.70 AKR1B1 (0.44) PNMTADRA2AADRA2BADRA2CMAPT
SCHEMBL429310 0.69 MAPT (0.57) PNMTADRA2AADRA2BADRA2CMAPT
SCHEMBL15656347 0.69 NR3C2 (0.39) PNMTADRA2AADRA2BADRA2CMAPT
SCHEMBL15497921 0.68 ALDH1A1 (0.44) PNMTADRA2AADRA2BADRA2CMAPT
Hydrochloric Acid SCHEMBL4967505 0.68 MAPT (0.56) PNMTADRA2AADRA2BADRA2CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1971604-A2 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF CANCER DISEASES Amgen Inc. (US) 2008-09-24 EP disclosed
WO-2007048070-A2 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF CANCER DISEASES AMGEN INC. (US) 2007-04-26 WO disclosed
EP-1697361-A1 BICYCLOHETEROARYLAMINE COMPOUNDS AS ION CHANNEL LIGANDS AND USES THEREOF Renovis, Inc. (US) 2006-09-06 EP disclosed
WO-2005066171-A1 BICYCLOHETEROARYLAMINE COMPOUNDS AS ION CHANNEL LIGANDS AND USES THEREOF RENOVIS, INC. (US) 2005-07-21 WO disclosed