SCHEMBL4017459

SCHEMBL4017459

O=CCC1CCc2ccc([N+](=O)[O-])cc2N1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PNMT P11086 8/20 0.42
ADRA2A P08913 5/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
GRIN2B Q13224 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2484227 0.79 CMA1 (0.39) PNMTADRA2AADRA2BADRA2C
SCHEMBL2776785 0.78 PNMT (0.43) PNMTADRA2AADRA2BADRA2CGRIN2B
SCHEMBL4970728 0.78 PNMT (0.40) PNMTADRA2AADRA2BADRA2C
SCHEMBL4429953 0.76 PNMT (0.52) PNMTADRA2AADRA2BADRA2CGRIN2B
SCHEMBL13233996 0.75 GRIN2B (0.42) PNMTADRA2AADRA2BADRA2CGRIN2B
SCHEMBL6195263 0.75 SIRT2 (0.45) PNMTADRA2AADRA2BADRA2CGRIN2B
SCHEMBL7456470 0.74 PNMT (0.56) PNMTADRA2AADRA2BADRA2CGRIN2B
SCHEMBL6197463 0.74 PNMT (0.54) PNMTADRA2AADRA2BADRA2CGRIN2B
SCHEMBL28439970 0.74 ALDH1A1 (0.41) PNMTADRA2AADRA2BADRA2C
SCHEMBL8702101 0.72 GRIN2B (0.42) PNMTADRA2AADRA2BADRA2CGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009089042-A1 PYRAZOLE PYRAZINE AMINE COMPOUNDS AS KINASE INHIBITORS, COMPOSITIONS THEREOF AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2009-07-16 WO disclosed