SCHEMBL4972425

SCHEMBL4972425

O=C(O)N1CCCC(C(Br)c2cccc(F)c2)C1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.41
DPP7 Q9UHL4 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
REN P00797 5/20 0.40
SCD5 Q86SK9 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HTT P42858 1/20 0.40
CHRM3 P20309 3/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4975348 0.86 DPP4 (0.42) DPP4DPP7KDM4EALDH1A1HPGD
SCHEMBL4975353 0.86 DPP4 (0.42) DPP4DPP7KDM4EALDH1A1HPGD
SCHEMBL3607883 0.83 GPR119 (0.48) REN
SCHEMBL3607879 0.83 GPR119 (0.48) REN
SCHEMBL4974370 0.80 REN (0.41) DPP4DPP7KDM4EALDH1A1HPGD
SCHEMBL4974097 0.79 REN (0.53) REN
SCHEMBL4978806 0.79 REN (0.53) REN
SCHEMBL4970186 0.78 REN (0.55) REN
SCHEMBL4970187 0.78 REN (0.55) REN
SCHEMBL4246324 0.75 REN (0.51) ALDH1A1HPGDSMN1; SMN2RENKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed