SCHEMBL497318

SCHEMBL497318

CC(C)(C)OC(=O)N1CCO[C@@H](c2ccc(OCCCBr)cc2)C1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 14/20 0.45
POLB P06746 1/20 0.40
RAB9A P51151 1/20 0.40
PDE4B Q07343 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL497356 0.87 HRH3 (0.56) POLB
SCHEMBL497233 0.85 HRH3 (0.43) POLBRAB9A
SCHEMBL28767928 0.84 POLB (0.43) GPR119POLBRAB9APDE4B
SCHEMBL503532 0.82 RORC (0.49) PDE4B
SCHEMBL1993504 0.82 RORC (0.49) PDE4B
SCHEMBL503531 0.82 RORC (0.49) PDE4B
SCHEMBL323889 0.81 USP2 (0.46) GPR119PDE4B
SCHEMBL497161 0.81 USP2 (0.46) GPR119PDE4B
SCHEMBL1438341 0.80 ALDH1A1 (0.43) GPR119POLB
SCHEMBL503547 0.80 NR1H2 (0.45) GPR119RAB9APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106045-B2 2-morpholino-4-pyrimidone compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-01-31 US disclosed
CN-101035781-A 2-morpholino-4-pyrimidone compound MITSUBISHI PHARMA CORP (JP) 2007-09-12 CN disclosed