SCHEMBL4974841

SCHEMBL4974841

Cc1ccc(Cl)cc1C(O)C1CCCN(C(=O)O)C1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 2/20 0.40
PROKR1 Q8TCW9 10/20 0.40
RAB9A P51151 1/20 0.39
TSHR P16473 1/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 1/20 0.38
ALOX12 P18054 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4974838 1.00 KMT2A (0.40) KMT2AALDH1A1MEN1PROKR1RAB9A
SCHEMBL2327230 0.85 CNR1 (0.46) KMT2AALDH1A1MEN1RAB9AMAPT
SCHEMBL2327223 0.85 CNR1 (0.46) KMT2AALDH1A1MEN1RAB9AMAPT
SCHEMBL2327226 0.85 CNR1 (0.46) KMT2AALDH1A1MEN1RAB9AMAPT
SCHEMBL28779404 0.83 KDM4E (0.42) KMT2AMEN1HTTSMN1; SMN2
SCHEMBL3963369 0.81 TSHR (0.41) KMT2AALDH1A1MEN1RAB9ATSHR
SCHEMBL4974885 0.78 TSHR (0.42) KMT2AALDH1A1MEN1PROKR1TSHR
SCHEMBL4974880 0.78 TSHR (0.42) KMT2AALDH1A1MEN1PROKR1TSHR
SCHEMBL4193014 0.78 REN (0.59)
SCHEMBL4193008 0.78 REN (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed