SCHEMBL4975205

SCHEMBL4975205

C[C@H]1CN(CCc2cc(F)cc(F)c2F)CCN1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
XIAP P98170 6/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
KCNH2 Q12809 2/20 0.38
RIPK1 Q13546 1/20 0.35
BIRC2 Q13490 6/20 0.35
PARP1 P09874 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
SLC6A3 Q01959 1/20 0.35
MLNR O43193 9/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2022959 0.86 XIAP (0.40) XIAPPARP1PARP2MLNRCYP3A4
SCHEMBL20317464 0.80 SLC6A3 (0.43) XIAPSLC6A2SLC6A4KCNH2BIRC2
SCHEMBL3144417 0.74 MLNR (0.50) XIAPSLC6A2SLC6A4KCNH2SLC6A3
SCHEMBL3137966 0.74 MLNR (0.50) XIAPSLC6A2SLC6A4KCNH2SLC6A3
SCHEMBL3137952 0.74 MLNR (0.50) XIAPSLC6A2SLC6A4KCNH2SLC6A3
SCHEMBL20317594 0.73 SLC6A3 (0.58) SLC6A2SLC6A4KCNH2SLC6A3MLNR
SCHEMBL4574566 0.73 SIGMAR1 (0.40) RIPK1MLNRCYP3A4
SCHEMBL4590115 0.73 SIGMAR1 (0.40) RIPK1MLNRCYP3A4
SCHEMBL4590022 0.72 XIAP (0.48) XIAPMLNRCYP3A4
SCHEMBL3172097 0.72 KDM4E (0.55) XIAPMLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134036-A1 ALPHA-SUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-α]PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed