SCHEMBL4590115

SCHEMBL4590115

C[C@@H]1CN(Cc2cc(F)cc(F)c2F)C[C@@H](C)N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.40
RIPK1 Q13546 3/20 0.39
MLNR O43193 8/20 0.35
CYP3A4 P08684 2/20 0.34
KDM4E B2RXH2 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTR2B P41595 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4574566 1.00 SIGMAR1 (0.40) SIGMAR1RIPK1MLNRCYP3A4KDM4E
SCHEMBL2022959 0.84 XIAP (0.40) MLNRCYP3A4
SCHEMBL4573907 0.81 RIPK1 (0.36) RIPK1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL4574124 0.77 RIPK1 (0.37) RIPK1HTR2A
SCHEMBL4574119 0.74 RIPK1 (0.36) RIPK1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL4590891 0.74 SIGMAR1 (0.43) SIGMAR1RIPK1
SCHEMBL4975205 0.73 XIAP (0.39) RIPK1MLNRCYP3A4
SCHEMBL4574455 0.72 KDM4E (0.44) SIGMAR1KDM4ESMN1; SMN2MEN1ALDH1A1
SCHEMBL4590377 0.72 MLNR (0.42) RIPK1MLNRKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4574348 0.71 GRM2 (0.41) RIPK1MLNRKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed