SCHEMBL4980244

SCHEMBL4980244

O=C(O)c1cnc(-c2ccccc2)n1-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 6/20 0.44
TSHR P16473 2/20 0.44
HTT P42858 3/20 0.42
KDM4E B2RXH2 1/20 0.42
AVPR1A P37288 1/20 0.41
PI4KA P42356 1/20 0.41
PI4K2B Q8TCG2 1/20 0.41
PI4K2A Q9BTU6 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
GAA P10253 2/20 0.41
MDM2 Q00987 1/20 0.40
CYP2C19 P33261 3/20 0.40
NOTUM Q6P988 1/20 0.40
CYP1A2 P05177 2/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5353171 0.87 ADORA2A (0.43) SMN1; SMN2ALDH1A1TSHRHTTKDM4E
SCHEMBL16040506 0.81 ALDH1A1 (0.45) ALDH1A1TSHRHTTAVPR1AMEN1
SCHEMBL461803 0.79 HTT (0.49) SMN1; SMN2ALDH1A1TSHRHTTKDM4E
SCHEMBL4879878 0.79 AVPR1A (0.49) SMN1; SMN2ALDH1A1HTTKDM4EAVPR1A
SCHEMBL11978680 0.78 MEN1 (0.50) SMN1; SMN2ALDH1A1TSHRHTTKDM4E
SCHEMBL2225245 0.77 HPGDS (0.50) ALDH1A1KDM4EKMT2ACYP1A2MAPT
SCHEMBL4879887 0.75 COMT (0.49) SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL7062228 0.74 AVPR1A (0.50) SMN1; SMN2ALDH1A1TSHRKDM4EAVPR1A
SCHEMBL9960592 0.73 RECQL (0.34) SMN1; SMN2ALDH1A1TSHRKDM4EGAA
SCHEMBL3441565 0.73 ALDH1A1 (0.42) ALDH1A1TSHRHTTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984355-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION Takeda Pharmaceutical Company Limited (JP) 2008-10-29 EP disclosed
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed