SCHEMBL4983

SCHEMBL4983

C[C@]12CCC(=O)C=C1CC[C@@H]1[C@@H]2[C@@H](O)C[C@@]2(C)[C@H]1CC[C@]2(O)C(=O)CS

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 10/20 0.84
NR3C1 P04150 8/20 0.84
SMN1; SMN2 Q16637 3/20 0.84
CYP2C19 P33261 2/20 0.84
HSD17B10 Q99714 2/20 0.84
PGR P06401 2/20 0.84
SERPINA6 P08185 2/20 0.84
CYP3A4 P08684 2/20 0.84
NFKB1 P19838 2/20 0.84
MAPT P10636 2/20 0.84
SHBG P04278 1/20 0.84
NR3C2 P08235 1/20 0.84
KMT2A Q03164 1/20 0.84
LMNA P02545 2/20 0.78
AR P10275 1/20 0.77
CHRM1 P11229 1/20 0.77
PMP22 Q01453 1/20 0.69
TSHR P16473 1/20 0.69
POLB P06746 1/20 0.68
GAA P10253 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19327149 1.00 HIF1A (0.84) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
SCHEMBL5488066 1.00 HIF1A (0.84) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
Hydrocortisone SCHEMBL19465688 0.91 HIF1A (1.00) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
SCHEMBL22476662 0.91 HIF1A (0.85) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
Hydrocortisone SCHEMBL1560948 0.91 HIF1A (1.00) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
Hydrocortisone SCHEMBL24900238 0.91 HIF1A (1.00) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
Hydrocortisone SCHEMBL6932400 0.91 HIF1A (1.00) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
SCHEMBL14513165 0.91 HIF1A (0.85) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
Hydrocortisone SCHEMBL143923 0.91 HIF1A (1.00) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10
Hydrocortisone SCHEMBL1688689 0.91 HIF1A (1.00) HIF1ANR3C1SMN1; SMN2CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7364 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4739293-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF AUTOIMMUNE DISORDERS AZURA OPHTHALMICS LTD (IL) 2026-05-13 EP claimed
EP-4739291-A2 ADMINISTRATION OF KERATOLYTICS TO OCULAR AND PERIOCULAR SURFACES AZURA OPHTHALMICS LTD (IL) 2026-05-13 EP claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
WO-2026041906-A1 SEMI-SOLID PHARMACEUTICAL COMPOSITION MICRO-DISPENSER Azura Ophthalmics Ltd. (IL) 2026-02-26 WO claimed
EP-4301343-B1 PHARMACEUTICAL COMPOSITIONS WITH REDUCED SIDE EFFECT AND METHODS OF USING THE SAME TLC BIOPHARMACEUTICALS INC (US) 2025-11-19 EP claimed
US-20250322925-A1 METHODS OF MANAGING EOSINOPHILIC ESOPHAGITIS ELLODI PHARMACEUTICALS L P (US) 2025-10-16 US claimed
EP-4616867-A1 COMBINATION OF ENDOTHELIN RECEPTOR ANTAGONIST AND GLUCOCORTICOID FOR TREATING IGA NEPHROPATHY Sanreno Therapeutics (Shanghai) Limited (CN) 2025-09-17 EP claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-12377144-B2 Methods of treating cancer using multi-specific binding proteins that bind NKG2D, CD16 and a tumor-associated antigen DRAGONFLY THERAPEUTICS, INC. (US) 2025-08-05 US claimed
EP-4590313-A1 COMBINATION THERAPIES WITH ONCOLYTIC ADENOVIRUS AND TOPOISOMERASE I INHIBITORS OR PRODRUGS THEREOF Theriva Biologics, S.L. (ES) 2025-07-30 EP claimed
EP-0913154-A1 Antipsoriatic nail lacquer Hoechst Marion Roussel Deutschland GmbH (DE) 1999-05-06 EP claimed
EP-0904266-A1 NITROSATED AND NITROSYLATED COMPOUNDS AND COMPOSITIONS AND THEIR USE FOR TREATING RESPIRATORY DISORDERS Nitromed, Inc. (US) 1999-03-31 EP claimed
EP-0900233-A1 NOVEL STEROID NITRITE AND NITRATE ESTER DERIVATIVES USEFUL AS ANTI-INFLAMMATORY DRUGS G.D. SEARLE & CO. (US) 1999-03-10 EP claimed
CN-1198676-A Glucocorticold ehancement of gene expression RES DEV FOUDATION (US) 1998-11-11 CN claimed
WO-1998034595-A1 MEDICAL AEROSOL FORMULATIONS JAGO RESEARCH AG (CH) 1998-08-13 WO claimed
WO-1997041144-A1 NOVEL STEROID NITRITE AND NITRATE ESTER DERIVATIVES USEFUL AS ANTI-INFLAMMATORY DRUGS G.D. SEARLE & CO. (US) 1997-11-06 WO claimed
WO-1997034871-A1 NITROSATED AND NITROSYLATED COMPOUNDS AND COMPOSITIONS AND THEIR USE FOR TREATING RESPIRATORY DISORDERS NITROMED, INC. (US) 1997-09-25 WO claimed
WO-1997020578-A1 NON-PRESERVED TOPICAL CORTICOSTEROID FOR TREATMENT OF DRY EYE, FILAMENTARY KERATITIS, AND DELAYED TEAR CLEARANCE UNIVERSITY OF MIAMI (US) 1997-06-12 WO claimed
EP-0496520-A1 Novel bone acting agents MERCK & CO. INC. (US) 1992-07-29 EP claimed
US-4877781-A TIXOCORTOL PIVALATE, EPHEDRINE SULFATE, PRAMOXINE HYDROCHLORIDE; ANTIINFLAMMATORY AGENTS FOR HEMORRHOIDS LaHaye, Peter G. (US) 1989-10-31 US claimed