SCHEMBL5004063

SCHEMBL5004063

COC(=O)CN(C)c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HSD17B10 Q99714 2/20 0.46
POLB P06746 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
RAB9A P51151 3/20 0.44
PKM P14618 2/20 0.44
PTGS2 P35354 1/20 0.43
HDAC1 Q13547 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TSHR P16473 1/20 0.41
NR1D1 P20393 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32670823 0.84 CA12 (0.42) ALDH1A1SMN1; SMN2HSD17B10RAB9ATSHR
SCHEMBL8911970 0.84 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2HSD17B10POLBTDP1
SCHEMBL16980496 0.83 RAB9A (0.50) ALDH1A1SMN1; SMN2RAB9AL3MBTL1NPC1
Methyl Alcohol SCHEMBL28809124 0.82 CA12 (0.41) ALDH1A1SMN1; SMN2HSD17B10RAB9ATSHR
SCHEMBL28690878 0.82 MAPT (0.50) ALDH1A1SMN1; SMN2HSD17B10POLBRAB9A
SCHEMBL28791227 0.82 HPGD (0.46) ALDH1A1SMN1; SMN2POLBTDP1RAB9A
SCHEMBL5345206 0.81 POLB (0.44) ALDH1A1POLBTSHR
SCHEMBL10175567 0.81 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2HSD17B10POLBTDP1
SCHEMBL28791233 0.81 HPGD (0.45) ALDH1A1SMN1; SMN2POLBTDP1RAB9A
SCHEMBL29173926 0.80 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2RAB9AL3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118055930-A Thiadiazole derivative, composition and application thereof 北京丹擎医药科技有限公司 2024-05-17 CN disclosed
CN-117736104-A Method for synthesizing butanedicarboxylate derivative by visible light catalysis 常州大学 2024-03-22 CN disclosed
WO-2023061415-A1 THIADIAZOLYL DERIVATIVES, COMPOSITIONS AND USES THEREOF DANATLAS PHARMACEUTICALS CO., LTD. (CN) 2023-04-20 WO disclosed
WO-2023061415-A1 THIADIAZOLYL DERIVATIVES, COMPOSITIONS AND USES THEREOF DANATLAS PHARMACEUTICALS CO., LTD. (CN) 2023-04-20 WO disclosed
WO-2023060573-A1 NOVEL THIADIAZOLYL DERIVATIVES OF DNA POLYMERASE THETA INHIBITORS BEIJING DANATLAS PHARMACEUTICAL CO., LTD. (CN) 2023-04-20 WO disclosed
US-7414063-B2 Inhibitors of Akt (protein kinase B) ELI LILLY AND COMPANY (US) 2008-08-19 US disclosed
US-20070043040-A1 Inhibitors of akt (protein kinase b) ELI LILLY AND COMPANY 2007-02-22 US disclosed
EP-1611105-A1 ISOQUINOLINE-5-SULFONIC ACID AMIDES AS INHIBITORS OF AKT (PROTEIN KINASE B) ELI LILLY AND COMPANY (US) 2006-01-04 EP disclosed
WO-2004094386-A1 ISOQUINOLINE-5-SULFONIC ACID AMIDES AS INHIBITORS OF AKT (PROTEIN KINASE B) ELI LILLY AND COMPANY (US) 2004-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070043040-A1 Inhibitors of akt (protein kinase b) AKT1, AKT2, BRAF ALDH1A1 4411/4885SMN1; SMN2 2866/4885HSD17B10 2386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.