SCHEMBL5011675

SCHEMBL5011675

NC(c1ccc(-c2ccc(NC(=O)C3CC3)cc2)cc1)c1ccc(F)cc1F

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.47
KMT2A Q03164 5/20 0.47
NPSR1 Q6W5P4 1/20 0.44
MAPT P10636 2/20 0.43
HDAC3 O15379 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC2 Q92769 2/20 0.43
NAMPT P43490 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
TSHR P16473 1/20 0.41
MEN1 O00255 2/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 2/20 0.41
TP53 P04637 1/20 0.41
ABL1 P00519 1/20 0.40
GFER P55789 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011831 0.87 PTPN1 (0.48) PTPN1KMT2ANPSR1MAPTHDAC3
SCHEMBL5011271 0.76 PTPN1 (0.51) PTPN1KMT2ANPSR1MAPTNAMPT
SCHEMBL5014676 0.75 PTPN1 (0.56) PTPN1KMT2ANPSR1MAPTNAMPT
SCHEMBL14734057 0.73 KMT2A (0.78) PTPN1KMT2AMAPTNAMPTTSHR
Hydrochloric Acid SCHEMBL5794594 0.72 KMT2A (0.76) PTPN1KMT2AMAPTNAMPTTSHR
SCHEMBL4490301 0.71 HSD11B1 (0.43) HDAC3
SCHEMBL24251873 0.71 KMT2A (0.71) KMT2AL3MBTL1MEN1GAATP53
SCHEMBL12341489 0.71 NAMPT (0.51) KMT2ANPSR1MAPTNAMPTL3MBTL1
SCHEMBL5011692 0.71 PTPN1 (0.58) PTPN1KMT2ANPSR1MAPTNAMPT
SCHEMBL5009744 0.70 DHODH (0.50) PTPN1KMT2ANPSR1MAPTHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP disclosed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO disclosed