SCHEMBL5009844

SCHEMBL5009844

CC(O)Cc1ccc(-c2ccc(CC=O)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
MME P08473 8/20 0.37
ACE P12821 7/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
CPA1 P15085 2/20 0.36
ACE2 Q9BYF1 2/20 0.36
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
ACACB O00763 1/20 0.35
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1336531 0.85 ALDH1A1 (0.46) ALDH1A1CYP1A2CYP2D6MMEACE
SCHEMBL8719652 0.83 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2D6TP53TSHR
SCHEMBL3392101 0.78 HRH3 (0.43) TSHR
SCHEMBL196800 0.78 TAAR1 (0.48) TSHRADRB3AKR1C2
SCHEMBL8157608 0.78 TAAR1 (0.57) CYP2D6TSHRADRB1ADRB3
SCHEMBL8721457 0.78 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP2D6MMEACE
SCHEMBL4057353 0.77 PTGS1 (0.48) ALDH1A1TSHRADRB3MAPTAKR1C2
SCHEMBL21176913 0.77 TSHR (0.37) TP53TSHRADRB3AKR1C2
Hydrochloric Acid SCHEMBL21352581 0.76 HRH3 (0.41) ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL12002693 0.76 SIGMAR1 (0.42) ALDH1A1CYP1A2CYP2D6MMEGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP claimed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO claimed