SCHEMBL5010663

SCHEMBL5010663

CCOC(=O)C1CCN(C(N)=O)CC1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.68
ALDH1A1 P00352 7/20 0.64
GAA P10253 2/20 0.62
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
KDM4E B2RXH2 2/20 0.55
POLB P06746 1/20 0.55
CHRM1 P11229 1/20 0.53
MEN1 O00255 1/20 0.52
TSHR P16473 1/20 0.52
KMT2A Q03164 1/20 0.52
NPC1 O15118 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1981006 0.86 MAPT (0.64) MAPTALDH1A1GAACYP3A4CYP2D6
SCHEMBL14107690 0.86 MAPT (0.51) MAPTALDH1A1GAACYP3A4CYP2D6
Hydrochloric Acid SCHEMBL3765748 0.86 MAPT (0.64) MAPTALDH1A1GAACYP3A4CYP2D6
SCHEMBL1720494 0.85 MAPT (0.72) MAPTALDH1A1GAACYP3A4CYP2D6
SCHEMBL14081980 0.85 MAPT (0.50) MAPTALDH1A1GAACYP3A4CYP2D6
SCHEMBL5885563 0.84 MAPT (0.70) MAPTALDH1A1GAACYP3A4CYP2D6
SCHEMBL900124 0.84 MAPT (0.70) MAPTALDH1A1GAACYP3A4CYP2D6
Acetic Acid SCHEMBL17984593 0.83 MAPT (0.60) MAPTALDH1A1GAACYP3A4CYP2D6
SCHEMBL12297020 0.82 ALDH1A1 (0.69) MAPTALDH1A1GAACYP3A4CYP2D6
SCHEMBL6983298 0.82 MAPT (0.68) MAPTALDH1A1GAACYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1884513-A1 PYRAZOLE COMPOUND AND THERAPEUTIC AGENT FOR DIABETES COMPRISING THE SAME Japan Tobacco, Inc. (JP) 2008-02-06 EP claimed
US-20070032529-A1 Pyrazole compounds and their use as antidiabetes agents JAPAN TOBACCO INC. (JP) 2007-02-08 US claimed
CN-108341791-B Benzothiadiazole compound, preparation method and application thereof 中国科学院上海药物研究所 2020-09-29 CN disclosed
EP-1884513-A1 PYRAZOLE COMPOUND AND THERAPEUTIC AGENT FOR DIABETES COMPRISING THE SAME Japan Tobacco, Inc. (JP) 2008-02-06 EP disclosed
US-20070032529-A1 Pyrazole compounds and their use as antidiabetes agents JAPAN TOBACCO INC. (JP) 2007-02-08 US disclosed
WO-2001007409-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS ASTRAZENECA UK LIMITED (GB) 2001-02-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070032529-A1 Pyrazole compounds and their use as antidiabetes agents PYGL, GYS2, AGL MAPT 4621/4885ALDH1A1 1278/4885GAA 53/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.