SCHEMBL5010667

SCHEMBL5010667

CCOC(=O)CCN1CCN(c2ccccc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.61
HTR7 P34969 5/20 0.61
SIGMAR1 Q99720 5/20 0.60
TMEM97 Q5BJF2 4/20 0.60
SLC6A2 P23975 2/20 0.60
HRH2 P25021 2/20 0.60
HRH1 P35367 2/20 0.60
CHRM1 P11229 1/20 0.60
HRH3 Q9Y5N1 1/20 0.60
MAPT P10636 2/20 0.58
DRD2 P14416 1/20 0.58
DRD4 P21917 1/20 0.57
CHRM5 P08912 1/20 0.57
ADRA1D P25100 1/20 0.57
HTR1B P28222 1/20 0.57
HTR2A P28223 1/20 0.57
HTR2C P28335 1/20 0.57
HTR1E P28566 1/20 0.57
HTR2B P41595 1/20 0.57
SLC6A3 Q01959 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8160104 0.92 HTR1A (0.58) HTR1AHTR7SIGMAR1TMEM97SLC6A2
SCHEMBL11631677 0.87 MAPT (0.63) HTR1AHTR7SIGMAR1TMEM97SLC6A2
SCHEMBL11162215 0.87 KCNH2 (0.60) HTR1AHTR7SIGMAR1TMEM97SLC6A2
SCHEMBL6005398 0.86 HTR1A (0.59) HTR1ASIGMAR1TMEM97SLC6A2HRH2
SCHEMBL10763277 0.85 HTR1A (0.65) HTR1AHTR7MAPTHTR2AHTR2C
SCHEMBL20562281 0.85 HTR1A (0.64) HTR1AHTR7SIGMAR1MAPTDRD2
SCHEMBL14860445 0.85 ALDH1A1 (0.60) SIGMAR1MAPTDRD2CHRNA7
SCHEMBL23086717 0.85 ALDH1A1 (0.54) HTR1ASIGMAR1TMEM97SLC6A2HRH2
SCHEMBL3157629 0.85 KMT2A (0.68) HTR1AMAPTDRD2DRD4HTR2A
SCHEMBL6003242 0.85 KMT2A (0.54) HTR1ASIGMAR1TMEM97SLC6A2HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 99 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6001549-A IMAGING ELEMENT CONTAINING ANTISTATIC AGENT EASTMAN KODAK COMPANY (US) 1999-12-14 US claimed
US-5641967-A INCREASED PHOTOSTIMULATED LUMINESCENCE EASTMAN KODAK COMPANY (US) 1997-06-24 US claimed
WO-2008093920-A2 1,2-DIHYDRO-1-OXOPHTHALAZINYL DERIVATIVES HAVING BIOLOGICAL ACTIVITY ON SEROTONIN RECEPTORS 5-HT2A AND 5-HT2C, AND PREPARATION THEREOF DONGBU HITEK CO., LTD. (KR) 2008-08-07 WO disclosed
EP-1383772-B1 NITROGEN-BASED CAMPTOTHECIN DERIVATIVES CALIFORNIA PACIFIC MED CENTER (US) 2006-08-30 EP disclosed
CN-1246323-C Nitrogen-based camptothecin derivatives CALIFORNIA PACIFIC MED CENTER (US) 2006-03-22 CN disclosed
US-6933302-B2 Nitrogen-based homo-camptothecin derivatives CALIFORNIA PACIFIC MEDICAL CENTER (US) 2005-08-23 US disclosed
US-6855720-B2 Nitrogen-based camptothecin derivatives CALIFORNIA PACIFIC MEDICAL CENTER (US) 2005-02-15 US disclosed
US-6825207-B2 ANTICANCER AGENTS CALIFORNIA PACIFIC MEDICAL CENTER 2004-11-30 US disclosed
EP-1228124-B1 ELECTRICALLY CONDUCTIVE MICROGEL AND METHOD FOR PREPARING THE SAME Q SYS CO LTD (KR) 2004-11-03 EP disclosed
CN-1511159-A Nitrogen-based camptothecin derivatives ����������̫ƽ��ҽѧ���� 2004-07-07 CN disclosed
US-20040063740-A1 For treatment of cancer SUTTER WEST BAY HOSPITALS, DBA CALIFORNIA PACIFIC MEDICAL CENTER 2004-04-01 US disclosed
US-4214047-A Photographic elements having hydrophilic colloid layers containing hydrophobic addenda uniformly loaded in latex polymer particles EASTMAN KODAK COMPANY (US) 1980-07-22 US disclosed
US-4203716-A Photographic elements having hydrophilic colloid layers containing hydrophobic addenda uniformly loaded in latex polymer particles EASTMAN KODAK COMPANY (US) 1980-05-20 US disclosed
US-4199363-A Processes for achieving uniform, efficient distribution of hydrophobic materials through hydrophilic colloid layers and loaded latex compositions EASTMAN KODAK COMPANY (US) 1980-04-22 US disclosed
US-4193800-A COLOR DIFFUSION TRANSFER, POLYMER HAVING ACRYLOLAMINOPHENYL AMMONIUM UNITS KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1980-03-18 US disclosed
US-4133687-A Photographic elements having hydrophilic colloid layers containing compounds having activator precursors and hydrophobic developing agents uniformly loaded in latex polymer particles EASTMAN KODAK COMPANY (US) 1979-01-09 US disclosed
US-4092416-A Benzopyrone derivatives exhibiting anti-allergic activity BOEHRINGER MANNHEIM GMBH (DT) 1978-05-30 US disclosed
US-4070189-A CATIONIC POLYBENZYLVINYL AMMONIUM OR PHOSPHONIUM SALT EASTMAN KODAK COMPANY (US) 1978-01-24 US disclosed
US-4055429-A Inhibitor barrier layers for photographic materials EASTMAN KODAK COMPANY (US) 1977-10-25 US disclosed
US-3958995-A Photographic elements containing cross-linked mordants and processes of preparing said elements EASTMAN KODAK COMPANY (US) 1976-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063740-A1 For treatment of cancer MGMT, PAICS, DCK HTR1A 1728/4885HTR7 541/4885SIGMAR1 4740/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.