SCHEMBL5011879

SCHEMBL5011879

Cc1cc(C)cc(CN2C(=O)OC3(CCCCC3)N2C(=O)c2ccc(Br)cc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.38
KDM4E B2RXH2 2/20 0.38
GPR183 P32249 2/20 0.38
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
MEN1 O00255 3/20 0.36
POLB P06746 1/20 0.35
LMNA P02545 3/20 0.35
GAA P10253 3/20 0.35
MAPT P10636 3/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HPGD P15428 2/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CASP6 P55212 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5015165 0.76 ATM (0.47) KMT2AMEN1LMNAMAPTALDH1A1
SCHEMBL5011747 0.73 KCNK3 (0.40) KMT2AOPRM1OPRD1LMNAALDH1A1
SCHEMBL1086387 0.71 POLB (0.42) KMT2AGPR183MEN1POLBLMNA
SCHEMBL17077896 0.58 RAB9A (0.49) KMT2AOPRM1OPRD1LMNAGAA
SCHEMBL12812885 0.57 RAB9A (0.55) KMT2AMEN1LMNAMAPTALDH1A1
SCHEMBL24185725 0.55 HPGD (0.96) KMT2AMEN1POLBLMNAMAPT
SCHEMBL969583 0.55 HPGD (0.96) KMT2AMEN1POLBLMNAMAPT
SCHEMBL9366736 0.54 HPGD (0.49) KMT2AKDM4EALDH1A1HPGDTSHR
SCHEMBL971083 0.54 HPGD (1.00) KMT2AMEN1POLBLMNAMAPT
SCHEMBL644199 0.54 HPGD (0.92) KMT2AGPR183MEN1POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed