SCHEMBL5015165

SCHEMBL5015165

CC(=O)c1cccc(NC(=S)N2N(Cc3cc(C)cc(C)c3)C(=O)OC23CCCCC3)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.47
ALDH1A1 P00352 5/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ESR1 P03372 1/20 0.44
LMNA P02545 3/20 0.41
MAPT P10636 1/20 0.41
NPC1 O15118 5/20 0.41
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
STAT1 P42224 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4264555 0.76 ATM (0.52) ATMALDH1A1CYP3A4LMNAMAPT
SCHEMBL5011879 0.76 KMT2A (0.38) ALDH1A1NPSR1LMNAMAPTSMN1; SMN2
SCHEMBL5011747 0.70 KCNK3 (0.40) ALDH1A1CYP1A2CYP3A4LMNAHPGD
SCHEMBL5011835 0.70 CYP1A2 (0.43) ALDH1A1CYP1A2CYP3A4LMNAMAPT
SCHEMBL5456725 0.62 ALDH1A1 (0.83) ALDH1A1CYP1A2CYP3A4LMNAMAPT
SCHEMBL28879978 0.62 ALDH1A1 (0.72) ATMALDH1A1LMNAMAPTNPC1
SCHEMBL4102809 0.60 KMT2A (0.73) ALDH1A1CYP1A2NPSR1LMNAMAPT
SCHEMBL1884508 0.60 ALDH1A1 (0.73) ATMALDH1A1CYP1A2LMNAMAPT
SCHEMBL474709 0.59 KMT2A (0.70) ALDH1A1CYP1A2NPSR1LMNAMAPT
SCHEMBL5340030 0.59 MEN1 (0.89) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed